SCHEMBL8922476

SCHEMBL8922476

Clc1ccc(N2CCN(Cn3ncc4c3-c3ccccc3CC4)CC2)nc1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.44
MAPT P10636 1/20 0.44
DRD2 P14416 8/20 0.42
DRD4 P21917 7/20 0.42
DRD3 P35462 6/20 0.42
HTR7 P34969 4/20 0.40
SIGMAR1 Q99720 4/20 0.40
HTR1A P08908 3/20 0.40
HTR2A P28223 3/20 0.40
HTR2C P28335 3/20 0.40
TMEM97 Q5BJF2 3/20 0.40
KDM4E B2RXH2 1/20 0.38
GAA P10253 1/20 0.38
HSD17B10 Q99714 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
NAMPT P43490 1/20 0.38
SLC6A4 P31645 1/20 0.37
DRD1 P21728 2/20 0.37
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8923621 0.83 HTR3A (0.50) ALDH1A1DRD2DRD4DRD3HTR1A
SCHEMBL8921653 0.81 HRH3 (0.52) ALDH1A1DRD2HTR7HTR1AHTR2C
SCHEMBL8630532 0.76 DRD2 (0.46) ALDH1A1MAPTDRD2DRD4DRD3
SCHEMBL8924034 0.74 DRD3 (0.51) ALDH1A1MAPTDRD2DRD4DRD3
SCHEMBL1388980 0.72 DRD4 (0.48) ALDH1A1MAPTDRD2DRD4DRD3
SCHEMBL6927518 0.67 KDM4E (0.55) ALDH1A1MAPTDRD2DRD4DRD3
SCHEMBL6125262 0.65 KMT2A (0.58) DRD2DRD4DRD3HTR7SIGMAR1
SCHEMBL8924222 0.65 MAPT (0.47) ALDH1A1MAPTDRD2DRD4DRD3
SCHEMBL27507443 0.64 DRD2 (0.52) ALDH1A1MAPTDRD2DRD4DRD3
SCHEMBL1447393 0.64 CNR2 (0.55) ALDH1A1DRD2DRD4DRD3HTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5686480-A Fused tricyclic heteroaromatic derivatives as dopamine receptor subtype ligands MERCK, SHARP & DOHME, LTD. (GB) 1997-11-11 US claimed
US-5686480-A Fused tricyclic heteroaromatic derivatives as dopamine receptor subtype ligands MERCK, SHARP & DOHME, LTD. (GB) 1997-11-11 US disclosed