SCHEMBL8922507

SCHEMBL8922507

O=C(O)CCC(c1ccccc1)c1cccc(Cl)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASR P41180 1/20 0.52
MEN1 O00255 3/20 0.50
KMT2A Q03164 3/20 0.50
ACP3 P15309 1/20 0.49
CACNA2D1 P54289 2/20 0.46
CACNA1B Q00975 2/20 0.46
CACNB1 Q02641 2/20 0.46
CACNA1C Q13936 2/20 0.46
CACNA1G O43497 1/20 0.46
ALDH1A1 P00352 2/20 0.46
LMNA P02545 1/20 0.46
ALPL P05186 1/20 0.46
ALPI P09923 1/20 0.46
MAPT P10636 1/20 0.46
ALPG P10696 1/20 0.46
ALOX12 P18054 1/20 0.46
HTT P42858 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
IDO1 P14902 1/20 0.45
HPGD P15428 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28361247 0.97 KMT2A (0.49) CASRMEN1KMT2AACP3ALDH1A1
SCHEMBL13481005 0.84 TBXAS1 (0.58)
SCHEMBL3674189 0.84 CYP2D6 (0.54) ALDH1A1ALOX12HPGDCNR1
SCHEMBL8869652 0.83 MEN1 (0.56) CASRMEN1KMT2AACP3CACNA2D1
SCHEMBL9242975 0.82 SLC6A2 (0.44) CASRIDO1CNR1
SCHEMBL17814900 0.82 SLC6A2 (0.44) CASRIDO1CNR1
SCHEMBL27909941 0.82 ALDH1A1 (0.49) MEN1KMT2AACP3ALDH1A1HPGD
SCHEMBL20425537 0.82 KMT2A (0.46) CASRMEN1KMT2AACP3ALDH1A1
SCHEMBL5321437 0.82 SLC6A2 (0.44) CASRIDO1CNR1
SCHEMBL8921884 0.80 ACP3 (0.49) CASRACP3LMNAMAPTALOX12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5643904-A Substituted hexahdryoazepinones and tetrahydrobenzazepinones PFIZER INC. (US) 1997-07-01 US disclosed
EP-0625145-A1 3-PHENYLUREIDO-AZEPIN-2-ONES AND -BENZAZEPIN-2-ONES USEFUL AS CHOLECYSTOKININ ANTAGONISTS PFIZER INC. (US) 1994-11-23 EP disclosed
WO-1993015059-A1 3-PHENYLUREIDO-AZEPIN-2-ONES AND -BENZAZEPIN-2-ONES USEFUL AS CHOLECYSTOKININ ANTAGONISTS PFIZER INC. (US) 1993-08-05 WO disclosed