SCHEMBL8921884

SCHEMBL8921884

Cc1cccc(C(CCC(=O)O)c2ccccc2)c1

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ACP3 P15309 1/20 0.49
CYP19A1 P11511 3/20 0.47
SLC6A9 P48067 1/20 0.46
LMNA P02545 1/20 0.46
MAPT P10636 1/20 0.46
ALOX12 P18054 1/20 0.46
HTT P42858 1/20 0.46
MTNR1A P48039 3/20 0.44
MTNR1B P49286 3/20 0.44
CNR1 P21554 1/20 0.43
CNR2 P34972 1/20 0.43
MGAM O43451 1/20 0.43
GAA P10253 1/20 0.43
SI P14410 1/20 0.43
MGAM2 Q2M2H8 1/20 0.43
CASR P41180 1/20 0.42
TBXAS1 P24557 1/20 0.42
BRD4 O60885 1/20 0.42
FFAR1 O14842 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3674189 0.84 CYP2D6 (0.54) ALOX12MTNR1AMTNR1BCNR1CNR2
SCHEMBL15093694 0.83 ACP3 (0.45) ACP3SLC6A9FFAR1
SCHEMBL9152199 0.83 CTSA (0.52) ACP3SLC6A9LMNAMAPTMGAM
SCHEMBL9469383 0.82 ACP3 (0.44) ACP3SLC6A9FFAR1
SCHEMBL27491134 0.82 SLC6A9 (0.45) ACP3SLC6A9FFAR1
SCHEMBL4931341 0.82 SLC6A9 (0.45) ACP3SLC6A9FFAR1
SCHEMBL11838314 0.82 ACP3 (0.44) ACP3CYP19A1SLC6A9MAPTFFAR1
SCHEMBL27466804 0.81 CYP19A1 (0.50) ACP3CYP19A1SLC6A9LMNAMAPT
SCHEMBL8922507 0.80 CASR (0.52) ACP3LMNAMAPTALOX12HTT
SCHEMBL6301200 0.80 MTNR1A (0.67) LMNAMAPTALOX12HTTMTNR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5643904-A Substituted hexahdryoazepinones and tetrahydrobenzazepinones PFIZER INC. (US) 1997-07-01 US disclosed
US-5484917-A FOR TREATMENT AND PREVENTION OF GASTROINTESTINAL DISORDERS, PAIN AND ANXIETY PFIZER INC. (US) 1996-01-16 US disclosed
EP-0625145-A1 3-PHENYLUREIDO-AZEPIN-2-ONES AND -BENZAZEPIN-2-ONES USEFUL AS CHOLECYSTOKININ ANTAGONISTS PFIZER INC. (US) 1994-11-23 EP disclosed
WO-1993015059-A1 3-PHENYLUREIDO-AZEPIN-2-ONES AND -BENZAZEPIN-2-ONES USEFUL AS CHOLECYSTOKININ ANTAGONISTS PFIZER INC. (US) 1993-08-05 WO disclosed