SCHEMBL8923729

SCHEMBL8923729

CCOC(=O)COP(=O)(CN[C@@H](Cc1ccc(-c2ccccc2)cc1OC)C(=O)O)OCC(=O)OCC

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDCD1 Q15116 3/20 0.42
CD274 Q9NZQ7 3/20 0.42
PPARG P37231 3/20 0.38
PPARA Q07869 3/20 0.38
PPARD Q03181 2/20 0.38
ADRB1 P08588 1/20 0.37
ADRB3 P13945 1/20 0.37
MAPT P10636 3/20 0.37
KDM4E B2RXH2 2/20 0.37
HPGD P15428 2/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
ALDH1A1 P00352 2/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
ESR1 P03372 1/20 0.36
TP53 P04637 1/20 0.36
HSD17B10 Q99714 1/20 0.36
RECQL P46063 1/20 0.36
HTT P42858 1/20 0.35
EGFR P00533 1/20 0.35
KDR P35968 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7413312 0.84 MME (0.45)
SCHEMBL8924096 0.83 ADRB1 (0.36) PDCD1CD274PPARGPPARAADRB1
SCHEMBL8924065 0.83 ADRB1 (0.36) PDCD1CD274PPARGPPARAADRB1
SCHEMBL7411130 0.82 ITGA4 (0.42) PPARGPPARAMEN1KMT2A
SCHEMBL8921652 0.82 MME (0.45) POLBKMT2A
SCHEMBL8923043 0.82 ITGA4 (0.51)
SCHEMBL7413383 0.82 CD274 (0.44) PDCD1CD274PPARGPPARAPPARD
SCHEMBL7411493 0.82 MME (0.47) PDCD1CD274PPARGPPARAPPARD
SCHEMBL7411486 0.82 MME (0.47) PDCD1CD274PPARGPPARAPPARD
SCHEMBL8923722 0.77 PDCD1 (0.40) PDCD1CD274PPARGPPARAPPARD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0660840-B1 PHOSPHONO SUBSTITUTED TETRAZOLE DERIVATIVES CIBA GEIGY AG (CH) 1997-05-07 EP disclosed
US-5550119-A ENDOTHELIN-CONVERTING ENZYM INHIBITORS CIBA-GEIGY CORPORATION (US) 1996-08-27 US disclosed
EP-0660840-A1 PHOSPHONO SUBSTITUTED TETRAZOLE DERIVATIVES. CIBA GEIGY AG (CH) 1995-07-05 EP disclosed
WO-1994005677-A1 PHOSPHONO SUBSTITUTED TETRAZOLE DERIVATIVES CIBA-GEIGY AG (CH) 1994-03-17 WO disclosed