SCHEMBL8923783

SCHEMBL8923783

CC(C)(C)Nc1cccnc1N1CCN(C(=O)c2c[nH]c3ccc(N)cc23)CC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GFER P55789 1/20 0.42
ADRA2A P08913 1/20 0.40
ADORA3 P0DMS8 1/20 0.40
CHRM1 P11229 1/20 0.40
MAOA P21397 1/20 0.40
TBXA2R P21731 1/20 0.40
OPRM1 P35372 1/20 0.40
MDH1 P40925 1/20 0.40
KCNH2 Q12809 1/20 0.40
ABCG2 Q9UNQ0 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
GAA P10253 2/20 0.40
ALDH1A1 P00352 4/20 0.39
HSD17B10 Q99714 3/20 0.39
HPGD P15428 3/20 0.39
TNFSF11 O14788 2/20 0.38
TNF P01375 2/20 0.38
USP2 O75604 1/20 0.38
MAPK1 P28482 1/20 0.38
AVPR1A P37288 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9038015 0.89 ALDH1A1 (0.47) GFERADRA2AADORA3CHRM1MAOA
SCHEMBL5109661 0.88 ADRA2A (0.53) GFERADRA2AADORA3CHRM1MAOA
Hydrochloric Acid SCHEMBL9001495 0.88 ALDH1A1 (0.46) GFERADRA2AADORA3CHRM1MAOA
SCHEMBL9037637 0.88 GFER (0.56) GFERNPSR1GAAALDH1A1HPGD
SCHEMBL8985883 0.88 ALDH1A1 (0.50) GFERNPSR1ALDH1A1HSD17B10HPGD
Hydrochloric Acid SCHEMBL8985797 0.87 ALDH1A1 (0.49) GFERNPSR1ALDH1A1HSD17B10HPGD
SCHEMBL8922978 0.86 TNFSF11 (0.57) TNFSF11TNFKMT2AHTT
SCHEMBL8923153 0.84 TRPV1 (0.47) KCNH2NPSR1HSD17B10
SCHEMBL9038867 0.82 AVPR1A (0.43) GFERADRA2AADORA3CHRM1MAOA
SCHEMBL9037247 0.82 AVPR1A (0.43) GFERADRA2AADORA3CHRM1MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5599930-A Substituted indoles as anti-AIDS pharmaceuticals THE UPJOHN COMPANY (US) 1997-02-04 US disclosed
WO-1993001181-A1 SUBSTITUTED INDOLES AS ANTI-AIDS PHARMACEUTICALS THE UPJOHN COMPANY (US) 1993-01-21 WO disclosed