SCHEMBL8928250

SCHEMBL8928250

COc1cccc(CCCCNC(=O)C2CCCC2)c1

nearest known ligand 0.65

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 7/20 0.62
MTNR1B P49286 7/20 0.62
NQO2 P16083 1/20 0.55
KMT2A Q03164 1/20 0.54
ALDH1A1 P00352 2/20 0.53
HDAC1 Q13547 1/20 0.53
HDAC6 Q9UBN7 1/20 0.53
POLB P06746 1/20 0.53
PKM P14618 1/20 0.53
CYP3A4 P08684 1/20 0.53
CYP2C9 P11712 1/20 0.53
HSD17B10 Q99714 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8928075 0.98 MTNR1A (0.62) MTNR1AMTNR1BNQO2KMT2AALDH1A1
SCHEMBL8928078 0.95 MTNR1A (0.65) MTNR1AMTNR1BKMT2AHDAC1HDAC6
SCHEMBL8928226 0.91 MTNR1A (0.70) MTNR1AMTNR1BALDH1A1PKM
SCHEMBL5530350 0.83 ALDH1A1 (0.72) KMT2AALDH1A1POLBPKMCYP3A4
SCHEMBL8928132 0.81 MTNR1A (0.92) MTNR1AMTNR1BKMT2AHDAC1HDAC6
SCHEMBL8928103 0.79 MTNR1A (0.69) MTNR1AMTNR1BKMT2AHDAC1HDAC6
SCHEMBL8928088 0.79 MTNR1A (0.92) MTNR1AMTNR1BHDAC1HDAC6
SCHEMBL31036087 0.78 MTNR1A (0.90) MTNR1AMTNR1BHDAC1HDAC6
SCHEMBL8928131 0.78 MTNR1A (0.68) MTNR1AMTNR1BKMT2AHDAC1HDAC6
SCHEMBL8928133 0.78 MTNR1A (0.67) MTNR1AMTNR1BNQO2KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5541228-A Melatonergic agents BRISTOL-MYERS SQUIBB CO. (US) 1996-07-30 US claimed
EP-0706994-A1 Melatonergic agents BRISTOL-MYERS SQUIBB COMPANY (US) 1996-04-17 EP claimed
US-5661185-A AN ALKOXYPHENYL-ALKYLUREA COMPOUND TREATING SLEEP DISORDER BRISTOL-MYERS SQUIBB CO. (US) 1997-08-26 US disclosed
US-5541228-A Melatonergic agents BRISTOL-MYERS SQUIBB CO. (US) 1996-07-30 US disclosed
EP-0706994-A1 Melatonergic agents BRISTOL-MYERS SQUIBB COMPANY (US) 1996-04-17 EP disclosed