SCHEMBL8929550

SCHEMBL8929550

c1nc(Cc2ccc3[nH]ccc3c2)c2cc[nH]c2n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 1/20 0.42
CYP11B1 P15538 1/20 0.42
CYP11B2 P19099 1/20 0.42
EGFR P00533 3/20 0.41
KDR P35968 1/20 0.40
FLT1 P17948 1/20 0.39
PIK3CA P42336 1/20 0.39
PIK3CG P48736 1/20 0.39
MAP3K11 Q16584 3/20 0.39
TTBK1 Q5TCY1 2/20 0.39
TTBK2 Q6IQ55 2/20 0.39
CDC7 O00311 1/20 0.38
DBF4 Q9UBU7 1/20 0.38
LMNA P02545 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
AKT2 P31751 2/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
CYP3A4 P08684 2/20 0.38
CYP2D6 P10635 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8930212 0.79 DAO (0.42) EGFRKDRCDC7DBF4AKT2
SCHEMBL8929582 0.76 CDC7 (0.57) EGFRKDRFLT1TTBK1TTBK2
SCHEMBL8928889 0.76 JAK3 (0.42) TTBK1TTBK2CDC7DBF4AKT2
SCHEMBL8929547 0.75 CDC7 (0.42) TTBK1TTBK2CDC7DBF4AKT2
SCHEMBL8930219 0.71 SMYD3 (0.41) KDRMAP3K11
SCHEMBL6950768 0.71 CYP17A1 (0.39) CYP17A1CYP11B1CYP11B2EGFRKDR
SCHEMBL7021509 0.70 EGFR (0.70) EGFRKDRFLT1TTBK1TTBK2
SCHEMBL24345975 0.70 AKT2 (0.50) TTBK1TTBK2CDC7DBF4AKT2
SCHEMBL2598740 0.69 CYP17A1 (0.42) CYP17A1CYP11B1CYP11B2CYP2D6
Hydrochloric Acid SCHEMBL7020471 0.69 EGFR (0.69) EGFRKDRFLT1TTBK1TTBK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0795556-A1 4-Substituted pyrrolopyrimidine compounds as tyrosin kinase inhibitors PHARMACIA & UPJOHN S.p.A. (IT) 1997-09-17 EP claimed
EP-0795556-A1 4-Substituted pyrrolopyrimidine compounds as tyrosin kinase inhibitors PHARMACIA & UPJOHN S.p.A. (IT) 1997-09-17 EP disclosed