SCHEMBL8928889

SCHEMBL8928889

c1nc(Cc2ccc3c(c2)CCC3)c2cc[nH]c2n1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
JAK3 P52333 6/20 0.42
JAK2 O60674 2/20 0.42
JAK1 P23458 2/20 0.42
MPO P05164 1/20 0.39
AXL P30530 2/20 0.38
HPGDS O60760 1/20 0.38
AKT2 P31751 1/20 0.38
GSK3B P49841 1/20 0.38
PDE5A O76074 1/20 0.37
TTBK1 Q5TCY1 2/20 0.37
TTBK2 Q6IQ55 2/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
CDC7 O00311 1/20 0.36
DBF4 Q9UBU7 1/20 0.36
TYK2 P29597 1/20 0.36
BMX P51813 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7834633 0.79 MPO (0.42) MPOPDE5A
SCHEMBL8930219 0.77 SMYD3 (0.41)
SCHEMBL8929550 0.76 CYP17A1 (0.42) JAK2AKT2GSK3BTTBK1TTBK2
SCHEMBL8929582 0.74 CDC7 (0.57) JAK3JAK2JAK1TTBK1TTBK2
SCHEMBL20752219 0.74 JAK2 (0.58) JAK3JAK2JAK1AXLGSK3B
SCHEMBL7821656 0.74 MPO (0.37) MPOPDE5A
SCHEMBL7834634 0.74 AKT2 (0.40) MPOAKT2CDC7DBF4
SCHEMBL8929547 0.73 CDC7 (0.42) JAK3JAK2JAK1AXLAKT2
SCHEMBL8929209 0.72 EGFR (0.63) TTBK1TTBK2
SCHEMBL8930212 0.72 DAO (0.42) AXLAKT2CDC7DBF4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0795556-A1 4-Substituted pyrrolopyrimidine compounds as tyrosin kinase inhibitors PHARMACIA & UPJOHN S.p.A. (IT) 1997-09-17 EP claimed
EP-0795556-A1 4-Substituted pyrrolopyrimidine compounds as tyrosin kinase inhibitors PHARMACIA & UPJOHN S.p.A. (IT) 1997-09-17 EP disclosed