SCHEMBL8931146

SCHEMBL8931146

COc1ccc(OC)c(CNCC(N)(c2ccccc2)c2ccccc2)c1

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HIF1A Q16665 1/20 0.48
APLNR P35414 1/20 0.48
HTR2A P28223 2/20 0.47
KMT2A Q03164 2/20 0.47
HTR2C P28335 1/20 0.47
MEN1 O00255 1/20 0.47
IDO1 P14902 2/20 0.47
ADRA1A P35348 1/20 0.47
TAAR1 Q96RJ0 1/20 0.47
HTT P42858 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
ALDH1A1 P00352 2/20 0.44
HSD17B10 Q99714 1/20 0.44
KDM4E B2RXH2 1/20 0.44
TP53 P04637 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9229255 0.89 APLNR (0.63) APLNRHTR2AKMT2AHTR2CMEN1
Hydrochloric Acid SCHEMBL8931145 0.88 APLNR (0.61) APLNRHTR2AKMT2AHTR2CMEN1
SCHEMBL9351069 0.87 ADRA1A (0.51) HTR2AKMT2AHTR2CMEN1IDO1
SCHEMBL8931156 0.84 MEN1 (0.58) KMT2AMEN1ALDH1A1KDM4ETP53
Hydrochloric Acid SCHEMBL8931155 0.83 MEN1 (0.57) KMT2AMEN1SMN1; SMN2ALDH1A1KDM4E
SCHEMBL2900357 0.76 HTT (0.58) KMT2AMEN1HTTSMN1; SMN2ALDH1A1
SCHEMBL10032817 0.75 HTR2A (0.62) HTR2AKMT2AHTR2CMEN1SMN1; SMN2
SCHEMBL14299916 0.75 APLNR (0.61) APLNRHTR2AKMT2AHTR2CMEN1
SCHEMBL9351081 0.74 CYP2D6 (0.54) KMT2AMEN1ADRA1AHTTALDH1A1
SCHEMBL2891401 0.73 HTT (0.46) KMT2AMEN1HTTSMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2614408-B2 1997-05-28 JP claimed
WO-1993010073-A1 ACYCLIC ETHYLENEDIAMINE DERIVATIVES AS SUBSTANCE P RECEPTOR ANTAGONISTS PFIZER INC. (US) 1993-05-27 WO claimed
US-5521220-A Acyclic ethylenediamine derivatives PFIZER INC. (US) 1996-05-28 US disclosed
EP-0613458-A1 ACYCLIC ETHYLENEDIAMINE DERIVATIVES AS SUBSTANCE P RECEPTOR ANTAGONISTS PFIZER INC. (US) 1994-09-07 EP disclosed
WO-1993010073-A1 ACYCLIC ETHYLENEDIAMINE DERIVATIVES AS SUBSTANCE P RECEPTOR ANTAGONISTS PFIZER INC. (US) 1993-05-27 WO disclosed