SCHEMBL893147

SCHEMBL893147

O=C(O)NCCC(O)CCc1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.50
DPP4 P27487 1/20 0.49
MMP2 P08253 1/20 0.49
MMP9 P14780 1/20 0.49
MMP12 P39900 1/20 0.49
MMP13 P45452 1/20 0.49
MMP14 P50281 1/20 0.49
LMNA P02545 1/20 0.48
PKM P14618 1/20 0.48
MMP8 P22894 3/20 0.47
CNR2 P34972 1/20 0.46
CA12 O43570 1/20 0.46
CA2 P00918 1/20 0.46
CA9 Q16790 1/20 0.46
CYP2C9 P11712 2/20 0.46
CYP2C19 P33261 2/20 0.46
KDM4E B2RXH2 1/20 0.46
CYP2D6 P10635 1/20 0.45
KMT2A Q03164 1/20 0.45
CNR1 P21554 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3510092 0.84 MMP2 (0.50) TSHRDPP4MMP2MMP9MMP12
SCHEMBL3507239 0.84 LAP3 (0.49) TSHRCYP2C9CYP2C19CYP2D6CNR1
SCHEMBL203278 0.81 ANPEP (0.47) TSHRDPP4LMNAPKMMMP8
SCHEMBL4799370 0.81 MMP2 (0.55) TSHRDPP4MMP2MMP9MMP12
Acetic Acid SCHEMBL7279901 0.80 TSHR (0.58) TSHRDPP4MMP2MMP9MMP12
Phenethylcarbamic Acid SCHEMBL249525 0.79 CA12 (0.68) MMP2MMP9CA12CA2CA9
SCHEMBL22412962 0.79 CYP2D6 (0.40) CNR2CYP2C19CYP2D6KMT2ACNR1
Phenethylcarbamic Acid SCHEMBL4459966 0.77 CA12 (0.66) MMP2MMP9CA12CA2CA9
Phenethylcarbamic Acid SCHEMBL28010696 0.77 CA12 (0.66) MMP2MMP9CA12CA2CA9
Phenethylcarbamic Acid SCHEMBL9718519 0.77 CA12 (0.66) MMP2MMP9CA12CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20130131085-A1 CYTOCHROME P450 OXIDASE INHIBITORS AND USES THEREOF ABBOTT LABORATORIES (US) 2013-05-23 US disclosed
US-20120083490-A1 CYTOCHROME P450 OXIDASE INHIBITORS AND USES THEREOF ABBOTT LABORATORIES (US) 2012-04-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120083490-A1 CYTOCHROME P450 OXIDASE INHIBITORS AND USES THEREOF CYP3A43, CYP3A5, POR TSHR 4236/4885DPP4 975/4885MMP2 344/4885
US-20130131085-A1 CYTOCHROME P450 OXIDASE INHIBITORS AND USES THEREOF CYP3A43, CYP3A5, POR TSHR 4236/4885DPP4 975/4885MMP2 344/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.