SCHEMBL8932007

SCHEMBL8932007

C=CCc1c(Cl)cc([N+](=O)[O-])c(Cl)c1Cl

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR35 Q9HC97 2/20 0.43
TDP1 Q9NUW8 2/20 0.42
VCAM1 P19320 5/20 0.39
TSHR P16473 4/20 0.39
ALDH1A1 P00352 4/20 0.39
CYP3A4 P08684 3/20 0.39
HPGD P15428 1/20 0.39
ALOX15 P16050 1/20 0.39
HIF1A Q16665 1/20 0.39
TXNRD1 Q16881 1/20 0.39
TXNRD3 Q86VQ6 1/20 0.39
TXNRD2 Q9NNW7 1/20 0.39
MAPK1 P28482 1/20 0.37
GABRA1 P14867 1/20 0.33
GABRB2 P47870 1/20 0.33
KDM4A O75164 1/20 0.33
KDM4B O94953 1/20 0.33
CYP1A2 P05177 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10600640 0.87 TDP1 (0.42) GPR35TDP1VCAM1TSHRALDH1A1
SCHEMBL9251185 0.86 GPR35 (0.51) GPR35TDP1ALDH1A1CYP3A4HPGD
SCHEMBL30471243 0.77 GPR35 (0.47) GPR35TDP1VCAM1TSHRALDH1A1
SCHEMBL8411786 0.77 GPR35 (0.47) GPR35TDP1VCAM1TSHRALDH1A1
SCHEMBL31503783 0.74 GPR35 (0.43) GPR35TDP1VCAM1ALDH1A1CYP3A4
SCHEMBL10600459 0.73 TSHR (0.42) TSHRALDH1A1MAPK1
SCHEMBL10363810 0.72 GPR35 (0.44) GPR35TDP1VCAM1TSHRALDH1A1
SCHEMBL3650611 0.72 TDP1 (0.61) GPR35TDP1VCAM1TSHRALDH1A1
SCHEMBL29939725 0.72 TDP1 (0.61) GPR35TDP1VCAM1TSHRALDH1A1
SCHEMBL9282606 0.71 TSHR (0.42) GPR35TDP1VCAM1TSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0175151-B1 2,4-DICHLORO-3-ALKYL-6-NITROPHENOLS AND PROCESS FOR THEIR PREPARATION BAYER AG (DE) 1989-01-18 EP claimed
US-4670608-A CATALYTIC CHLORINATION OF 1-ALKYL-4-NITROBENZENE BAYER AKTIENGESELLSCHAFT (DE) 1987-06-02 US claimed
EP-0175151-A1 2,4-Dichloro-3-alkyl-6-nitrophenols and process for their preparation BAYER AG (DE) 1986-03-26 EP claimed
JP-9268158-A None JP disclosed
JP-9268158-A None JP disclosed
JP-9268159-A None JP disclosed
JP-9268159-A None JP disclosed
JP-H09268158-A PRODUCTION OF 3-ALKYL-6-NITRO-1,2,4-TRICHLOROBENZENE COMPOUND FUJI PHOTO FILM CO LTD 1997-10-14 JP disclosed
JP-H09268159-A PRODUCTION OF 3-ALKYL-6-NITRO-1,2,4-TRICHLOROBENZENE COMPOUND FUJI PHOTO FILM CO LTD 1997-10-14 JP disclosed
JP-H09268158-A PRODUCTION OF 3-ALKYL-6-NITRO-1,2,4-TRICHLOROBENZENE COMPOUND FUJI PHOTO FILM CO LTD 1997-10-14 JP disclosed
JP-H09268159-A PRODUCTION OF 3-ALKYL-6-NITRO-1,2,4-TRICHLOROBENZENE COMPOUND FUJI PHOTO FILM CO LTD 1997-10-14 JP disclosed
EP-0473464-B1 Process for preparing 2-4-dichloro-3-alkyl-6-nitrophenols TAOKA CHEMICAL CO LTD (JP) 1995-06-14 EP disclosed
US-5136109-A PROCESS FOR PREPARING 2,4-DICHLORO-3-ALKYL-6-NITROPHENOLS TAOKA CHEMICAL COMPANY, LTD. (JP) 1992-08-04 US disclosed
EP-0473464-A1 Process for preparing 2-4-dichloro-3-alkyl-6-nitrophenols TAOKA CHEMICAL CO., LTD (JP) 1992-03-04 EP disclosed
US-5012015-A Nitrading a trichlorobenzene with mixed acid, hydrolysis DAIEI CHEMICAL CO., LTD. (JP) 1991-04-30 US disclosed
EP-0175151-B1 2,4-DICHLORO-3-ALKYL-6-NITROPHENOLS AND PROCESS FOR THEIR PREPARATION BAYER AG (DE) 1989-01-18 EP disclosed
US-4670608-A CATALYTIC CHLORINATION OF 1-ALKYL-4-NITROBENZENE BAYER AKTIENGESELLSCHAFT (DE) 1987-06-02 US disclosed
EP-0175151-A1 2,4-Dichloro-3-alkyl-6-nitrophenols and process for their preparation BAYER AG (DE) 1986-03-26 EP disclosed