SCHEMBL8933213

SCHEMBL8933213

CC(C)(C)OC(=O)NCC(=O)N1CCC[C@]1(C(=O)O)C1CCCCC1.NC(=O)c1ccc(NC(=O)O)nc1

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 1/20 0.36
NAMPT P43490 1/20 0.35
EPHX2 P34913 1/20 0.35
MEN1 O00255 1/20 0.34
ALDH1A1 P00352 1/20 0.34
TSHR P16473 1/20 0.34
KMT2A Q03164 1/20 0.34
OPRM1 P35372 2/20 0.33
OPRK1 P41145 1/20 0.33
NPC1L1 Q9UHC9 3/20 0.33
OPRL1 P41146 1/20 0.33
BCL2 P10415 1/20 0.33
SIGMAR1 Q99720 1/20 0.33
NPFFR1 Q9GZQ6 1/20 0.33
NPFFR2 Q9Y5X5 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6489531 0.91 NPFFR1 (0.35) MEN1ALDH1A1TSHRKMT2AOPRM1
SCHEMBL6477215 0.88 JAK2 (0.37) NAMPTOPRM1OPRK1SIGMAR1NPFFR1
Acetic Acid SCHEMBL6477357 0.87 F2 (0.33) MEN1ALDH1A1TSHRKMT2ANPC1L1
SCHEMBL7705663 0.86 OPRM1 (0.32) MEN1ALDH1A1TSHRKMT2AOPRM1
SCHEMBL5900915 0.82 MEN1 (0.44) MEN1ALDH1A1TSHRKMT2ANPC1L1
SCHEMBL8781179 0.80 DPP4 (0.37)
SCHEMBL6485866 0.79 ITGB3 (0.33) OPRM1OPRK1
SCHEMBL6476534 0.78 JAK2 (0.36) OPRM1OPRK1
SCHEMBL5900918 0.77 MEN1 (0.45) MEN1ALDH1A1TSHRKMT2ASIGMAR1
SCHEMBL6482023 0.77 FAP (0.30) OPRM1OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996025426-A1 NOVEL DIPEPTIDE AMIDINES AS THROMBIN INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 1996-08-22 WO disclosed