SCHEMBL7705663

SCHEMBL7705663

CC(C)(C)OC(=O)NCC(=O)N1CCC[C@]1(C(=O)O)C1CCCCC1.COC(=O)NC(=N)c1ccc(C(N)=O)cn1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 1/20 0.32
OPRK1 P41145 1/20 0.32
F2 P00734 1/20 0.31
MMP1 P03956 1/20 0.31
MMP9 P14780 1/20 0.31
MMP13 P45452 1/20 0.31
STING1 Q86WV6 1/20 0.31
SIGMAR1 Q99720 1/20 0.31
NPFFR1 Q9GZQ6 1/20 0.31
NPFFR2 Q9Y5X5 1/20 0.31
NPC1L1 Q9UHC9 4/20 0.31
KLK5 Q9Y337 1/20 0.30
CKS1B P61024 1/20 0.30
SKP1 P63208 1/20 0.30
SKP2 Q13309 1/20 0.30
CHEK2 O96017 1/20 0.30
ELANE P08246 1/20 0.30
FAP Q12884 1/20 0.30
MEN1 O00255 1/20 0.30
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6489531 0.92 NPFFR1 (0.35) OPRM1OPRK1STING1SIGMAR1NPFFR1
Acetic Acid SCHEMBL6477357 0.91 F2 (0.33) F2SIGMAR1NPFFR1NPFFR2NPC1L1
SCHEMBL6477218 0.89 OPRK1 (0.33) OPRM1OPRK1
SCHEMBL6476916 0.87 OPRM1 (0.31) OPRM1OPRK1
SCHEMBL8933213 0.86 GRIN2B (0.36) OPRM1OPRK1SIGMAR1NPFFR1NPFFR2
SCHEMBL6477215 0.84 JAK2 (0.37) OPRM1OPRK1SIGMAR1NPFFR1NPFFR2
SCHEMBL6482023 0.84 FAP (0.30) OPRM1OPRK1FAP
SCHEMBL8725919 0.83
SCHEMBL6485866 0.83 ITGB3 (0.33) OPRM1OPRK1F2FAP
SCHEMBL8781179 0.81 DPP4 (0.37)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6444817-B1 ANTICOAGULANTS ABBOTT LABORATORIES 2002-09-03 US disclosed
US-6030972-A 2- OR 5-AMINOMETHYL,2- OR 5-CYANOPYRIMIDINES AS INTERMEDIATES OF ANTICOAGULANTS IN EXTRACORPOREAL CIRCULATION (HEART-LUNG MACHINE, HEMODIALYSIS) BASF AKTIENGESELLSCHAFT (DE) 2000-02-29 US disclosed
EP-0873356-A1 NOVEL DIPEPTIDE AMIDINES AS THROMBIN INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 1998-10-28 EP disclosed
WO-1996025426-A1 NOVEL DIPEPTIDE AMIDINES AS THROMBIN INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 1996-08-22 WO disclosed