SCHEMBL8933349

SCHEMBL8933349

N=C(NO)c1ccc(C(N)=O)cn1.O=C(C=NCC(=O)N1CCC[C@]1(C(=O)O)C1CCCCC1)OCc1ccccc1

nearest known ligand 0.34

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
FKBP1A P62942 2/20 0.33
HDAC3 O15379 2/20 0.33
HDAC1 Q13547 2/20 0.33
HDAC2 Q92769 2/20 0.33
HDAC6 Q9UBN7 2/20 0.33
OPRK1 P41145 2/20 0.32
KCNH2 Q12809 1/20 0.32
OPRM1 P35372 1/20 0.31
CHRNB2 P17787 1/20 0.30
CHRNA7 P36544 1/20 0.30
CHRNA4 P43681 1/20 0.30
ACHE P22303 2/20 0.30
PRKAB2 O43741 1/20 0.30
PRKAG1 P54619 1/20 0.30
PRKAA2 P54646 1/20 0.30
PRKAA1 Q13131 1/20 0.30
PRKAG3 Q9UGI9 1/20 0.30
PRKAG2 Q9UGJ0 1/20 0.30
PRKAB1 Q9Y478 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8933077 0.88
SCHEMBL8725919 0.84
SCHEMBL8933278 0.84 OPRK1 (0.32) OPRK1KCNH2
SCHEMBL8725915 0.81 OPRM1 (0.30) OPRK1OPRM1
SCHEMBL8725715 0.78 ITGB3 (0.34)
SCHEMBL6482023 0.77 FAP (0.30) OPRK1OPRM1
SCHEMBL8933238 0.75 ITGB3 (0.31)
SCHEMBL6477218 0.75 OPRK1 (0.33) OPRK1KCNH2OPRM1
SCHEMBL6487745 0.73 ITGB3 (0.36) HDAC6OPRK1KCNH2OPRM1PRKAA2
SCHEMBL6476916 0.72 OPRM1 (0.31) OPRK1OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996025426-A1 NOVEL DIPEPTIDE AMIDINES AS THROMBIN INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 1996-08-22 WO disclosed