SCHEMBL8933479

SCHEMBL8933479

CCOC(=O)c1nc2ccsc2nc1N.CCOC(=O)c1nc2ccsc2nc1NCc1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 4/20 0.53
CYP1A2 P05177 1/20 0.53
CYP3A4 P08684 1/20 0.53
GAA P10253 1/20 0.53
CYP2C9 P11712 1/20 0.53
CYP2C19 P33261 1/20 0.53
MEN1 O00255 3/20 0.51
KMT2A Q03164 3/20 0.51
SMN1; SMN2 Q16637 5/20 0.50
ALDH1A1 P00352 4/20 0.47
MAPT P10636 3/20 0.47
CDC7 O00311 1/20 0.46
DBF4 Q9UBU7 1/20 0.46
HSD17B10 Q99714 2/20 0.45
KDM4E B2RXH2 1/20 0.45
SLC26A6 Q9BXS9 2/20 0.44
RAB9A P51151 2/20 0.43
PDE4A P27815 1/20 0.43
PDE4B Q07343 1/20 0.43
PDE4C Q08493 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8144214 0.95 NPSR1 (0.58) NPSR1CYP1A2CYP3A4GAACYP2C9
SCHEMBL8128482 0.84 ALDH1A1 (0.46) NPSR1CYP1A2CYP3A4GAACYP2C9
SCHEMBL8137173 0.81 NPSR1 (0.40) NPSR1CYP1A2CYP3A4GAACYP2C9
SCHEMBL2840279 0.80 NPSR1 (0.73) NPSR1CYP1A2CYP3A4GAACYP2C9
SCHEMBL8139117 0.78 CDC7 (0.43) NPSR1CYP1A2CYP2C9MEN1KMT2A
SCHEMBL8127687 0.78 LMNA (0.41) NPSR1CYP1A2CYP3A4GAACYP2C9
SCHEMBL8143187 0.77 MAPK8 (0.42) NPSR1CYP1A2CYP3A4GAACYP2C9
SCHEMBL13510962 0.76 NPSR1 (0.67) NPSR1CYP1A2CYP3A4GAACYP2C9
SCHEMBL8144240 0.75 NPC1 (0.37) NPSR1CYP1A2CYP2C9MEN1KMT2A
SCHEMBL24261170 0.75 ADORA2A (0.68) NPSR1MEN1KMT2ARAB9AADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996022992-A1 TRICYCLIC SUBSTITUTED HEXAHYDROBENZ[E]ISOINDOLE ALPHA-1 ADRENERGIC ANTAGONISTS ABBOTT LABORATORIES (US) 1996-08-01 WO disclosed