SCHEMBL8936429

SCHEMBL8936429

Cn1c(NC(=O)NCc2ccccc2)c(-c2ccc(F)cc2)c2c(F)cccc2c1=O

nearest known ligand 0.61

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 7/20 0.61
ALDH1A1 P00352 6/20 0.46
KDM4E B2RXH2 4/20 0.46
LMNA P02545 3/20 0.46
HPGD P15428 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
POLB P06746 2/20 0.46
NPC1 O15118 1/20 0.46
MAOB P27338 1/20 0.46
RAB9A P51151 1/20 0.46
KMT2A Q03164 2/20 0.45
L3MBTL1 Q9Y468 1/20 0.44
RORC P51449 1/20 0.43
MEN1 O00255 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8936601 0.89 TACR1 (0.70) TACR1ALDH1A1KDM4ELMNAHPGD
SCHEMBL8936542 0.84 TACR1 (0.86) TACR1ALDH1A1KDM4ELMNAHPGD
SCHEMBL8936576 0.76 TACR1 (1.00) TACR1ALDH1A1KDM4EHPGDSMN1; SMN2
SCHEMBL8785120 0.75 TACR1 (0.45) TACR1ALDH1A1KDM4ELMNASMN1; SMN2
SCHEMBL8936577 0.73 TACR1 (0.76) TACR1ALDH1A1KMT2AMEN1
SCHEMBL8936508 0.72 TACR1 (0.59) TACR1ALDH1A1KDM4EHPGDPOLB
SCHEMBL8936439 0.72 TACR1 (0.86) TACR1SMN1; SMN2NPC1RAB9AKMT2A
SCHEMBL8936527 0.71 TACR1 (0.90) TACR1ALDH1A1KDM4EHPGDSMN1; SMN2
SCHEMBL9178393 0.71 TACR1 (0.57) TACR1KDM4ESMN1; SMN2POLBNPC1
SCHEMBL8936587 0.71 TACR1 (0.64) TACR1ALDH1A1KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5523305-A ANALGESICS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-06-04 US disclosed
EP-0566069-A1 Tachykinin receptor antagonists, isoquinolones and their production TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-10-20 EP disclosed