SCHEMBL8936579

SCHEMBL8936579

C=CCN1C(=O)c2ccccc2Oc2nc(Cl)ccc21

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 1/20 0.44
ALDH1A1 P00352 8/20 0.41
MAPT P10636 5/20 0.41
LMNA P02545 4/20 0.41
PKM P14618 1/20 0.41
GALR3 O60755 1/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
TDP1 Q9NUW8 2/20 0.40
CRHBP P24387 1/20 0.40
MAPK1 P28482 1/20 0.40
CRHR2 Q13324 1/20 0.40
POLB P06746 3/20 0.38
RXFP1 Q9HBX9 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
HDAC3 O15379 2/20 0.36
TUBB4A P04350 2/20 0.36
TUBB P07437 2/20 0.36
TUBA3C P0DPH7 2/20 0.36
HDAC4 P56524 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8936624 0.81 HDAC3 (0.40) ALDH1A1MAPTLMNAPOLBSMN1; SMN2
SCHEMBL8936600 0.79 HDAC3 (0.43) CASP3ALDH1A1MAPTLMNAMEN1
SCHEMBL9101209 0.73 TP53 (0.54) CASP3ALDH1A1MAPTLMNAPKM
SCHEMBL8936617 0.71 NR1H2 (0.33) ALDH1A1HDAC3TUBB4ATUBBTUBA3C
SCHEMBL8936654 0.69 TP53 (0.45) ALDH1A1MAPTLMNAKMT2APOLB
SCHEMBL8936648 0.69 TP53 (0.45) ALDH1A1MAPTLMNAKMT2APOLB
SCHEMBL31377051 0.68 CASP3 (0.85) CASP3ALDH1A1MAPTLMNAPKM
SCHEMBL170913 0.68 CASP3 (0.85) CASP3ALDH1A1MAPTLMNAPKM
SCHEMBL4901773 0.68 CTSG (0.40) CASP3ALDH1A1MAPTLMNAMEN1
SCHEMBL8936630 0.68 TP53 (0.51) MAPTLMNAMEN1KMT2APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5547951-A ENZYME INHIBITORS; AIDS BOEHRINGER INGELHEIM PHARAMCEUTICALS, INC. (US) 1996-08-20 US disclosed
EP-0417534-A1 Pyrido[2,3-b][1,4]benzoxazepin (and thiazepin)-6(5H)-ones and thiones and their use in the prevention or treatment of AIDS Boehringer Ingelheim Pharmaceuticals Inc. (US) 1991-03-20 EP disclosed