SCHEMBL8936654

SCHEMBL8936654

CC=CCN1C(=O)c2ccccc2Oc2ncccc21

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.45
MAPT P10636 3/20 0.40
LMNA P02545 2/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
POLB P06746 2/20 0.39
KMT2A Q03164 1/20 0.38
HDAC3 O15379 1/20 0.38
TUBB4A P04350 1/20 0.38
TUBB P07437 1/20 0.38
TUBA3C P0DPH7 1/20 0.38
HDAC4 P56524 1/20 0.38
TUBA1B P68363 1/20 0.38
TUBA4A P68366 1/20 0.38
TUBB4B P68371 1/20 0.38
TUBB3 Q13509 1/20 0.38
HDAC1 Q13547 1/20 0.38
TUBB2A Q13885 1/20 0.38
TUBB8 Q3ZCM7 1/20 0.38
TUBA3E Q6PEY2 1/20 0.38
TUBA1A Q71U36 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8936648 1.00 TP53 (0.45) TP53MAPTLMNASMN1; SMN2POLB
SCHEMBL9853427 0.79 TP53 (0.48) TP53MAPTLMNASMN1; SMN2POLB
SCHEMBL8936730 0.79 TP53 (0.53) TP53MAPTPOLBKMT2AALDH1A1
SCHEMBL8936630 0.77 TP53 (0.51) TP53MAPTLMNAPOLBKMT2A
SCHEMBL9853429 0.77 NR1H2 (0.47) TP53MAPTLMNASMN1; SMN2POLB
SCHEMBL9101209 0.76 TP53 (0.54) TP53MAPTLMNASMN1; SMN2POLB
SCHEMBL9101435 0.74 TP53 (0.60) TP53MAPTLMNASMN1; SMN2POLB
SCHEMBL8936669 0.72 TP53 (0.46) TP53MAPTLMNASMN1; SMN2POLB
SCHEMBL8936588 0.72 MAPT (0.50) MAPTLMNASMN1; SMN2POLBKMT2A
SCHEMBL9212981 0.72 TP53 (0.58) TP53MAPTLMNASMN1; SMN2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5547951-A ENZYME INHIBITORS; AIDS BOEHRINGER INGELHEIM PHARAMCEUTICALS, INC. (US) 1996-08-20 US disclosed
EP-0417534-A1 Pyrido[2,3-b][1,4]benzoxazepin (and thiazepin)-6(5H)-ones and thiones and their use in the prevention or treatment of AIDS Boehringer Ingelheim Pharmaceuticals Inc. (US) 1991-03-20 EP disclosed