SCHEMBL8936741

SCHEMBL8936741

Cn1nnc2ccc(Sc3ccc(Cl)cc3Cn3cncn3)cc21

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 8/20 0.46
CYP11B1 P15538 2/20 0.46
KDM4E B2RXH2 2/20 0.40
POLB P06746 1/20 0.40
HTT P42858 1/20 0.40
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
CCR1 P32246 1/20 0.35
CCR2 P41597 1/20 0.35
CCR4 P51679 1/20 0.35
FAAH O00519 1/20 0.35
SLC6A4 P31645 1/20 0.33
F2 P00734 1/20 0.33
F10 P00742 1/20 0.33
LRRK2 Q5S007 3/20 0.33
ALDH1A1 P00352 1/20 0.33
HPGD P15428 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8936772 0.80 CYP19A1 (0.47) CYP19A1CYP11B1CCR1CCR2CCR4
SCHEMBL8936722 0.78 CYP19A1 (0.46) CYP19A1CYP11B1MEN1KMT2ACCR1
SCHEMBL9201316 0.76 CYP19A1 (0.46) CYP19A1CYP11B1CCR1CCR2CCR4
SCHEMBL8936793 0.75 CCR1 (0.40) CYP19A1KDM4EPOLBHTTMEN1
SCHEMBL8936764 0.74 NLRP3 (0.40) CYP19A1CYP11B1KDM4EMEN1KMT2A
SCHEMBL8936743 0.71 PDE7A (0.43) KDM4EPOLBHTTMEN1KMT2A
SCHEMBL8710156 0.69 CYP19A1 (0.43) CYP19A1CYP11B1KDM4EPOLBHTT
SCHEMBL8936729 0.68 CYP19A1 (0.41) CYP19A1CYP11B1KDM4EMEN1KMT2A
SCHEMBL14476937 0.68 KEAP1 (0.53) CYP19A1CYP11B1KDM4EMEN1KMT2A
SCHEMBL8936731 0.67 NLRP3 (0.39) CYP19A1CYP11B1CCR1CCR2CCR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5587392-A THERAPY FOR ESTROGEN DEPENDENT DISEASES MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1996-12-24 US disclosed
EP-0684235-A1 Novel azolyl methyl phenyl derivatives having aromatase inhibitory activity MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1995-11-29 EP disclosed