SCHEMBL8938342

SCHEMBL8938342

O=C(O)c1[nH]c2ccc(Cl)cc2c1[S+]([O-])c1ccccc1

nearest known ligand 0.58

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAP2 P11137 4/20 0.58
ALDH1A1 P00352 2/20 0.46
KDM4E B2RXH2 1/20 0.46
POLB P06746 4/20 0.46
MAPT P10636 3/20 0.44
PKM P14618 1/20 0.44
LMNA P02545 1/20 0.44
THRB P10828 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
CYP1A2 P05177 1/20 0.44
HPGD P15428 1/20 0.44
XBP1 P17861 1/20 0.44
CYP2C19 P33261 1/20 0.44
PTGS2 P35354 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8938249 0.90 MAP2 (0.60) MAP2ALDH1A1KDM4EPOLBMAPT
SCHEMBL9034407 0.84 ALDH1A1 (0.64) MAP2ALDH1A1KDM4EMAPTLMNA
SCHEMBL8938321 0.83 PTGS2 (0.52) MAP2ALDH1A1KDM4EPOLBMAPT
SCHEMBL8938413 0.79 CNR1 (0.45) ALDH1A1KDM4EPOLBPTGS2
SCHEMBL9033744 0.77 MAPK3 (0.43) MAP2ALDH1A1KDM4EPOLBPTGS2
SCHEMBL9040770 0.76 MCL1 (0.44) MAP2ALDH1A1KDM4EPOLBMAPT
SCHEMBL9032423 0.75 PTGS2 (0.50) MAP2ALDH1A1KDM4EPOLBMAPT
SCHEMBL8938478 0.75 PTGS2 (0.42) MAP2ALDH1A1KDM4EPOLBMAPT
SCHEMBL6921821 0.74 MAP2 (0.65) MAP2ALDH1A1KDM4EPOLBLMNA
SCHEMBL42364 0.73 MAP2 (1.00) MAP2ALDH1A1KDM4EPOLBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5527819-A TREATING AIDS MERCK & CO., INC. (US) 1996-06-18 US disclosed
EP-0686148-A4 INHIBITORS OF HIV REVERSE TRANSCRIPTASE MERCK & CO INC (US) 1996-02-07 EP disclosed
EP-0686148-A1 INHIBITORS OF HIV REVERSE TRANSCRIPTASE MERCK & CO. INC. (US) 1995-12-13 EP disclosed
WO-1994019321-A1 INHIBITORS OF HIV REVERSE TRANSCRIPTASE MERCK & CO., INC. (US) 1994-09-01 WO disclosed