SCHEMBL9033744

SCHEMBL9033744

O=C(NCc1ccnc(Cl)c1)c1[nH]c2ccc(Cl)cc2c1[S+]([O-])c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK3 P27361 1/20 0.43
MAPK1 P28482 1/20 0.43
CNR1 P21554 6/20 0.43
PTGS2 P35354 2/20 0.42
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
PPARG P37231 1/20 0.40
PPARD Q03181 1/20 0.40
PPARA Q07869 1/20 0.40
POLB P06746 1/20 0.39
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
EGFR P00533 1/20 0.38
NHERF1 O14745 1/20 0.38
MCL1 Q07820 1/20 0.38
MAP2 P11137 1/20 0.38
GABRP O00591 1/20 0.37
GABRD O14764 1/20 0.37
GABRA1 P14867 1/20 0.37
GABRB1 P18505 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8938413 0.90 CNR1 (0.45) MAPK3MAPK1CNR1PTGS2KDM4E
SCHEMBL8938478 0.81 PTGS2 (0.42) CNR1PTGS2KDM4EALDH1A1POLB
SCHEMBL8938242 0.79 TUBB4A (0.46) MAPK3MAPK1CNR1PTGS2KDM4E
SCHEMBL9032423 0.79 PTGS2 (0.50) CNR1PTGS2KDM4EALDH1A1PPARG
SCHEMBL9040770 0.78 MCL1 (0.44) CNR1PTGS2KDM4EALDH1A1POLB
SCHEMBL8938342 0.77 MAP2 (0.58) PTGS2KDM4EALDH1A1POLBMAP2
SCHEMBL8938321 0.75 PTGS2 (0.52) CNR1PTGS2KDM4EALDH1A1POLB
SCHEMBL8938249 0.75 MAP2 (0.60) MAPK1KDM4EALDH1A1POLBMAP2
SCHEMBL9034407 0.72 ALDH1A1 (0.64) PTGS2KDM4EALDH1A1MEN1KMT2A
SCHEMBL8938394 0.70 TUBB4A (0.45) CNR1PTGS2KDM4EALDH1A1PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0686148-A4 INHIBITORS OF HIV REVERSE TRANSCRIPTASE MERCK & CO INC (US) 1996-02-07 EP disclosed
EP-0686148-A1 INHIBITORS OF HIV REVERSE TRANSCRIPTASE MERCK & CO. INC. (US) 1995-12-13 EP disclosed