SCHEMBL8938478

SCHEMBL8938478

Cn1ccnc1CNC(=O)c1[nH]c2ccc(Cl)cc2c1[S+]([O-])c1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 3/20 0.42
CNR1 P21554 7/20 0.41
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
EGFR P00533 1/20 0.38
MAPT P10636 2/20 0.38
LMNA P02545 1/20 0.38
THRB P10828 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
SLC40A1 Q9NP59 1/20 0.38
POLB P06746 2/20 0.38
MAP2 P11137 1/20 0.37
USP1 O94782 1/20 0.37
CNR2 P34972 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8938413 0.82 CNR1 (0.45) PTGS2CNR1KDM4EALDH1A1POLB
SCHEMBL9033744 0.81 MAPK3 (0.43) PTGS2CNR1KDM4EALDH1A1EGFR
SCHEMBL8938368 0.80 TUBB4A (0.47) PTGS2CNR1KDM4EALDH1A1EGFR
SCHEMBL9032423 0.78 PTGS2 (0.50) PTGS2CNR1KDM4EALDH1A1EGFR
SCHEMBL8938331 0.76 TUBB4A (0.50) PTGS2CNR1SLC40A1CNR2
SCHEMBL8938321 0.75 PTGS2 (0.52) PTGS2CNR1KDM4EALDH1A1MAPT
SCHEMBL8938342 0.75 MAP2 (0.58) PTGS2KDM4EALDH1A1MAPTLMNA
SCHEMBL13859620 0.74 KDM4E (0.41) PTGS2CNR1KDM4EALDH1A1MAPT
SCHEMBL8938249 0.73 MAP2 (0.60) KDM4EALDH1A1MAPTLMNATHRB
SCHEMBL9040770 0.72 MCL1 (0.44) PTGS2CNR1KDM4EALDH1A1EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0686148-A4 INHIBITORS OF HIV REVERSE TRANSCRIPTASE MERCK & CO INC (US) 1996-02-07 EP claimed
EP-0686148-A1 INHIBITORS OF HIV REVERSE TRANSCRIPTASE MERCK & CO. INC. (US) 1995-12-13 EP claimed
WO-1994019321-A1 INHIBITORS OF HIV REVERSE TRANSCRIPTASE MERCK & CO., INC. (US) 1994-09-01 WO claimed
US-5527819-A TREATING AIDS MERCK & CO., INC. (US) 1996-06-18 US disclosed
EP-0686148-A4 INHIBITORS OF HIV REVERSE TRANSCRIPTASE MERCK & CO INC (US) 1996-02-07 EP disclosed
EP-0686148-A1 INHIBITORS OF HIV REVERSE TRANSCRIPTASE MERCK & CO. INC. (US) 1995-12-13 EP disclosed
WO-1994019321-A1 INHIBITORS OF HIV REVERSE TRANSCRIPTASE MERCK & CO., INC. (US) 1994-09-01 WO disclosed