SCHEMBL8938792

SCHEMBL8938792

Cc1ccc(CN2CCC(Oc3ccc4c(=O)[nH]cc(C)c4c3)CC2)c(Cl)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 1/20 0.51
OPRM1 P35372 4/20 0.46
OPRD1 P41143 2/20 0.46
OPRK1 P41145 2/20 0.46
CACNA1F O60840 1/20 0.46
CHRM2 P08172 1/20 0.46
CHRM1 P11229 1/20 0.46
DRD2 P14416 1/20 0.46
DRD1 P21728 1/20 0.46
DRD4 P21917 1/20 0.46
ADRA1D P25100 1/20 0.46
HTR7 P34969 1/20 0.46
ADRA1A P35348 1/20 0.46
ADRA1B P35368 1/20 0.46
DRD3 P35462 1/20 0.46
OPRL1 P41146 1/20 0.46
CACNA1D Q01668 1/20 0.46
CACNA1S Q13698 1/20 0.46
CACNA1C Q13936 1/20 0.46
MAOA P21397 4/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8935171 0.93 ROCK1 (0.51) ROCK1MAOAMAOBHRH1CCR3
SCHEMBL8935163 0.90 ROCK1 (0.52) ROCK1OPRM1MAOAMAOBHRH1
SCHEMBL8935224 0.87 ROCK1 (0.55) ROCK1MAOAMAOBHRH1CCR3
SCHEMBL8938824 0.87 OPRM1 (0.48) ROCK1OPRM1OPRD1OPRK1CACNA1F
SCHEMBL8938636 0.85 ROCK1 (0.53) ROCK1OPRM1OPRD1OPRK1CACNA1F
SCHEMBL8935147 0.84 MAOB (0.62) ROCK1MAOAMAOBHRH1CCR3
SCHEMBL8935217 0.83 ROCK1 (0.53) ROCK1MAOAMAOBHRH1CCR3
SCHEMBL8935195 0.83 MAOA (0.61) ROCK1OPRK1MAOAMAOBHRH1
SCHEMBL8938789 0.83 ROCK1 (0.51) ROCK1MAOAMAOBHRH1CCR3
SCHEMBL8938969 0.82 OPRM1 (0.44) OPRM1OPRD1OPRK1CACNA1FCHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8188117-B2 Piperidinyl-substituted isoquinolone derivatives SANOFI-AVENTIS (FR) 2012-05-29 US disclosed