SCHEMBL8938958

SCHEMBL8938958

Cc1c[nH]c(=O)c2ccc(OC3CCN(CCC(C)(F)F)CC3)c(F)c12

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 12/20 0.40
CCR3 P51677 12/20 0.40
KCNH2 Q12809 4/20 0.35
ROCK1 Q13464 1/20 0.34
HTR1A P08908 1/20 0.33
HTR7 P34969 1/20 0.33
NUAK1 O60285 1/20 0.33
MAOA P21397 1/20 0.32
MAOB P27338 1/20 0.32
S1PR5 Q9H228 1/20 0.32
PARP1 P09874 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8936592 0.93 HRH1 (0.40) HRH1CCR3KCNH2ROCK1HTR1A
SCHEMBL8939065 0.90 HTR1A (0.37) HRH1CCR3KCNH2HTR1AMAOA
SCHEMBL8936483 0.86 MAOA (0.46) HRH1CCR3KCNH2HTR1AMAOA
SCHEMBL8936493 0.86 HRH1 (0.42) HRH1CCR3KCNH2ROCK1MAOA
SCHEMBL8936546 0.85 HRH1 (0.42) HRH1CCR3KCNH2HTR1AHTR7
SCHEMBL8934493 0.85 MAOA (0.39) HRH1CCR3KCNH2ROCK1MAOA
SCHEMBL8938964 0.83 HRH1 (0.39) HRH1CCR3KCNH2MAOAMAOB
SCHEMBL8936533 0.83 HRH1 (0.46) HRH1CCR3KCNH2ROCK1
SCHEMBL8937203 0.83 HTR1A (0.37) HRH1CCR3KCNH2HTR1AMAOA
SCHEMBL8936820 0.82 ADRB2 (0.43) HRH1CCR3KCNH2MAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8188117-B2 Piperidinyl-substituted isoquinolone derivatives SANOFI-AVENTIS (FR) 2012-05-29 US disclosed