SCHEMBL8939062

SCHEMBL8939062

CCc1c[nH]c(=O)c2ccc(OC3CCN(Cc4cc(C)cc(Cl)c4)CC3)c(F)c12

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 6/20 0.41
CCR3 P51677 6/20 0.41
MAOA P21397 3/20 0.39
MAOB P27338 3/20 0.39
SCN1A P35498 1/20 0.38
SCN8A Q9UQD0 1/20 0.38
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
KCNH2 Q12809 1/20 0.37
SSTR5 P35346 2/20 0.36
POLB P06746 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8937216 0.96 HRH1 (0.42) HRH1CCR3MAOAMAOBSCN1A
SCHEMBL8938967 0.91 HRH1 (0.44) HRH1CCR3MAOAMAOBSCN1A
SCHEMBL8937220 0.89 HRH1 (0.39) HRH1CCR3MAOAMAOBSCN1A
SCHEMBL8937204 0.89 MAOA (0.49) HRH1CCR3MAOAMAOBSCN1A
SCHEMBL8936704 0.89 HRH1 (0.45) HRH1CCR3MAOAMAOBKCNH2
SCHEMBL13890296 0.88 ACHE (0.42) HRH1CCR3MAOAMAOBSCN1A
SCHEMBL8939080 0.84 HRH1 (0.39) HRH1CCR3MAOAMAOBSCN1A
SCHEMBL8937187 0.82 HRH1 (0.39) HRH1CCR3KCNH2
SCHEMBL8937219 0.82 OPRM1 (0.41) HRH1CCR3SCN1ASCN8AMEN1
SCHEMBL8937227 0.82 ACHE (0.43) CCR3SCN1ASCN8AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8188117-B2 Piperidinyl-substituted isoquinolone derivatives SANOFI-AVENTIS (FR) 2012-05-29 US disclosed