SCHEMBL8939734

SCHEMBL8939734

C=CCOc1ccc[c]c1Cc1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.41
TSHR P16473 1/20 0.41
MAPK1 P28482 1/20 0.41
HSD17B10 Q99714 1/20 0.41
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
LIG1 P18858 1/20 0.39
ALDH1A1 P00352 2/20 0.36
KDM4E B2RXH2 1/20 0.36
SLC22A1 O15245 1/20 0.35
LMNA P02545 1/20 0.35
CYP1A2 P05177 1/20 0.35
ADRB2 P07550 1/20 0.35
ADRB1 P08588 1/20 0.35
HTR1A P08908 1/20 0.35
CYP2D6 P10635 1/20 0.35
HTR2A P28223 1/20 0.35
SLC6A4 P31645 1/20 0.35
ADRA1A P35348 1/20 0.35
CA12 O43570 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8939743 0.81 MAPT (0.49) MAPK1HTR1ASLC6A4ADRA1AMAPT
SCHEMBL8939785 0.80 HTR1A (0.42) HPGDTSHRMAPK1HSD17B10MEN1
SCHEMBL27982817 0.80 TSHR (0.41) HPGDTSHRMAPK1HSD17B10LIG1
SCHEMBL8939792 0.76 CYP1A2 (0.46) HPGDTSHRLMNACYP1A2CYP3A4
SCHEMBL8859963 0.76 LTA4H (0.44) HPGDMEN1KMT2AHTR1ACYP2D6
SCHEMBL3849532 0.74 HPGD (0.44) HPGDTSHRMAPK1HSD17B10LIG1
SCHEMBL7687255 0.73 HTR2A (0.37) HPGDMEN1KMT2AKDM4ECYP1A2
SCHEMBL5889093 0.73 HPGD (0.44) HPGDTSHRMAPK1HSD17B10LIG1
SCHEMBL15068016 0.72 TSHR (0.42) HPGDTSHRMAPK1HSD17B10LIG1
SCHEMBL15068002 0.72 ALDH1A1 (0.43) HPGDTSHRMAPK1HSD17B10LIG1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5516797-A SUPPRESSING GRAFT REJECTION VERTEX PHARMACEUTICALS, INCORPORATED (US) 1996-05-14 US disclosed
US-5330993-A Immunosuppressive compounds VERTEX PHARMACEUTICALS, INC. (US) 1994-07-19 US disclosed