SCHEMBL8939839

SCHEMBL8939839

C[C@@H]1C[C@H](OC(=O)C(C)(C)C)[C@@]2(C)CC[C@H]3[C@@H](CC[C@H]4N(C)CCC[C@]34C)[C@H]12

nearest known ligand 0.38

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
AR P10275 1/20 0.33
KCNH2 Q12809 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8650498 0.82 SRD5A1 (0.48)
SCHEMBL8650495 0.82 SRD5A1 (0.48)
SCHEMBL8925259 0.73 AR (0.38) ARKCNH2KMT2A
SCHEMBL8925043 0.71 AR (0.39) ARKCNH2KMT2A
SCHEMBL9301232 0.71 SRD5A2 (0.54)
SCHEMBL8650483 0.71 SRD5A1 (0.35) KMT2A
SCHEMBL8651043 0.71 SRD5A1 (0.35) KMT2A
SCHEMBL8926885 0.69 SRD5A1 (0.43) ARKCNH2KMT2A
SCHEMBL9663769 0.68 SRD5A2 (0.42)
SCHEMBL8609868 0.68 CA2 (0.34) ARKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0700291-A4 15-SUBSTITUTED 4-AZASTEROIDS MERCK & CO INC (US) 1996-07-03 EP claimed
EP-0700291-A1 15-SUBSTITUTED 4-AZASTEROIDS MERCK & CO. INC. (US) 1996-03-13 EP claimed
WO-1994020104-A1 15-SUBSTITUTED 4-AZASTEROIDS MERCK & CO, INC. (US) 1994-09-15 WO claimed