SCHEMBL8941277

SCHEMBL8941277

COc1ccc(Cc2cnc(Cl)nc2Cl)cc1OC

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHFR P00374 1/20 0.59
HTT P42858 1/20 0.59
CA2 P00918 1/20 0.53
NTRK1 P04629 1/20 0.47
CSF1R P07333 1/20 0.47
NTRK3 Q16288 1/20 0.47
NTRK2 Q16620 1/20 0.47
PDE2A O00408 1/20 0.47
ABCC4 O15439 1/20 0.47
USP2 O75604 1/20 0.47
PDE5A O76074 1/20 0.47
ABCB11 O95342 1/20 0.47
ALDH1A1 P00352 1/20 0.47
LMNA P02545 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C9 P11712 1/20 0.47
ALOX15 P16050 1/20 0.47
TSHR P16473 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11863386 0.84 DHFR (0.58) DHFRALDH1A1CYP3A4TSHRNFKB1
SCHEMBL10847549 0.81 DHFR (0.42) DHFRHTTALDH1A1CYP3A4TSHR
SCHEMBL27407372 0.80 CA2 (0.67) DHFRHTTCA2PDE2AABCC4
SCHEMBL8549099 0.79 DHFR (0.60) DHFRHTT
SCHEMBL1748366 0.78 KDM4E (0.46) DHFRHTTALDH1A1SMN1; SMN2PDE10A
SCHEMBL8941118 0.75 DHFR (0.45) DHFRHTTALDH1A1LMNAACHE
Diaveridine SCHEMBL29527560 0.74 DHFR (1.00) DHFRHTTNTRK1CSF1RNTRK3
Diaveridine SCHEMBL93896 0.74 DHFR (1.00) DHFRHTTNTRK1CSF1RNTRK3
SCHEMBL12682418 0.73 CA2 (0.66) DHFRHTTCA2ALDH1A1LMNA
SCHEMBL10794425 0.73 PLA2G7 (0.43) LMNATSHRSMN1; SMN2PDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5491234-A Pyrimidine derivatives for enhancing antitumor activity PFIZER INC. (US) 1996-02-13 US disclosed
EP-0580753-B1 PYRIMIDINE DERIVATIVES FOR ENHANCING ANTITUMOR ACTIVITY PFIZER (US) 1995-03-01 EP disclosed