SCHEMBL8943779

SCHEMBL8943779

Nc1ccc(-c2ccccc2)cc1CC1NC(=O)NC1=O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADAMTS5 Q9UNA0 2/20 0.42
GAA P10253 2/20 0.40
IKBKB O14920 1/20 0.37
IDO1 P14902 1/20 0.35
MAPT P10636 3/20 0.35
CASP1 P29466 2/20 0.35
AURKA O14965 1/20 0.35
THRB P10828 1/20 0.35
TTK P33981 1/20 0.35
AURKB Q96GD4 1/20 0.35
INCENP Q9NQS7 1/20 0.35
ADAMTS4 O75173 1/20 0.34
CXCR4 P61073 1/20 0.34
ALDH1A1 P00352 3/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
KDM4E B2RXH2 1/20 0.34
USP2 O75604 1/20 0.34
LMNA P02545 1/20 0.34
HSP90AA1 P07900 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7389924 0.80 GAA (0.42) ADAMTS5GAAMAPTCASP1ADAMTS4
SCHEMBL10761843 0.79 GAA (0.37) GAAIDO1MAPTCASP1THRB
SCHEMBL12258527 0.78 HDAC8 (0.47) ADAMTS5GAACASP1ADAMTS4CXCR4
SCHEMBL18076579 0.78 TDP2 (0.43) ADAMTS5GAACXCR4MAOAMAOB
SCHEMBL7389935 0.71 MAPT (0.39) GAAMAPTALDH1A1LMNAHTT
SCHEMBL7390658 0.71 ADAMTS5 (0.39) ADAMTS5GAAHDAC1
SCHEMBL1011632 0.71 HDAC8 (0.57) ADAMTS5GAAADAMTS4CXCR4MAOB
SCHEMBL14357764 0.71 HDAC8 (0.57) ADAMTS5GAAADAMTS4CXCR4MAOB
SCHEMBL7883790 0.70 CXCR4 (0.40) ADAMTS5GAAIDO1CASP1THRB
SCHEMBL17111472 0.69 NTRK1 (0.45) ADAMTS5GAAMAPTCASP1ADAMTS4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5541325-A ENZYME INHIBITORS, ANTIALLERGENS JANSSEN PHARMACEUTICA N.V. (BE) 1996-07-30 US disclosed