SCHEMBL8945868

SCHEMBL8945868

CC1=Nc2ccccc2CC(c2cccs2)N1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
BCHE P06276 3/20 0.39
NOS2 P35228 3/20 0.38
NOS3 P29474 2/20 0.38
ALDH1A1 P00352 6/20 0.37
SLC6A2 P23975 1/20 0.35
SLC6A4 P31645 1/20 0.35
SLC6A3 Q01959 1/20 0.35
KDM4E B2RXH2 2/20 0.34
ACHE P22303 1/20 0.34
MEN1 O00255 2/20 0.33
MAPT P10636 2/20 0.33
KMT2A Q03164 2/20 0.33
GAA P10253 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
CYP2D6 P10635 1/20 0.33
RECQL P46063 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11149139 0.78 MAPT (0.47) BCHEALDH1A1KDM4EMEN1MAPT
SCHEMBL8945915 0.78 MEN1 (0.36) ALDH1A1KDM4EMEN1MAPTKMT2A
Hydrochloric Acid SCHEMBL9582485 0.77 MEN1 (0.46) BCHEALDH1A1KDM4EMEN1MAPT
SCHEMBL8945950 0.74 NOS2 (0.40) BCHENOS2NOS3ALDH1A1SLC6A2
SCHEMBL28923871 0.74 AR (0.45) NOS2NOS3ALDH1A1SLC6A2SLC6A4
SCHEMBL8945774 0.71 SLC6A2 (0.40) BCHENOS2NOS3ALDH1A1SLC6A2
SCHEMBL2376720 0.70 KDM4E (0.54) NOS2NOS3ALDH1A1KDM4EACHE
SCHEMBL8945814 0.67 GAA (0.44) BCHEALDH1A1KDM4EMEN1MAPT
SCHEMBL4053132 0.67 ALDH1A1 (0.46) ALDH1A1KDM4EMEN1MAPTKMT2A
SCHEMBL8945788 0.66 MEN1 (0.38) BCHENOS2NOS3ALDH1A1SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5510346-A ANTIDEPRESSANTS, ANTIANXIETY AGENTS HOECHST MARION ROUSSEL, INC. (US) 1996-04-23 US disclosed
US-5292760-A 4-heteroaryl-1,3-benzodiazepines and 2-substituted-α-(heteroaryl)benzeneethanamines HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-03-08 US disclosed
EP-0322582-A2 4-Heteroaryl-1,3-Benzodiazepines and 2-substituted-alpha-(heteroaryl)benzeneethanamines, a process for their preparation and their use us medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-07-05 EP disclosed