SCHEMBL8945915

SCHEMBL8945915

CC1=Nc2ccccc2CC(c2ccsc2)N1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.36
KMT2A Q03164 4/20 0.36
SMN1; SMN2 Q16637 4/20 0.36
KDM4E B2RXH2 2/20 0.36
MAPT P10636 2/20 0.36
HSD17B10 Q99714 1/20 0.36
ADORA2B P29275 5/20 0.34
GAA P10253 1/20 0.33
ALDH1A1 P00352 1/20 0.33
POLB P06746 1/20 0.33
CYP2D6 P10635 1/20 0.33
RECQL P46063 1/20 0.33
PKM P14618 1/20 0.32
PDE3B Q13370 1/20 0.32
PDE3A Q14432 1/20 0.32
LMNA P02545 2/20 0.31
OPRM1 P35372 3/20 0.31
OPRD1 P41143 2/20 0.31
OPRK1 P41145 2/20 0.31
HTT P42858 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11149139 0.84 MAPT (0.47) MEN1KMT2ASMN1; SMN2KDM4EMAPT
Hydrochloric Acid SCHEMBL9582485 0.82 MEN1 (0.46) MEN1KMT2ASMN1; SMN2KDM4EMAPT
SCHEMBL8945868 0.78 BCHE (0.39) MEN1KMT2AKDM4EMAPTGAA
SCHEMBL8945994 0.76 HSD17B10 (0.34) MEN1KMT2ASMN1; SMN2KDM4EMAPT
SCHEMBL8945923 0.70 HRH4 (0.35)
SCHEMBL8945925 0.70 ADORA2B (0.32) ADORA2BOPRM1OPRK1
SCHEMBL8946148 0.70 ADORA2B (0.33) MEN1KMT2ASMN1; SMN2KDM4EHSD17B10
Hydrochloric Acid SCHEMBL8945865 0.69 ADORA2B (0.32) MEN1KMT2ASMN1; SMN2ADORA2BLMNA
Hydrochloric Acid SCHEMBL8945921 0.69 HRH4 (0.34)
Hydrochloric Acid SCHEMBL8945951 0.69 ADORA2B (0.31) ADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5510346-A ANTIDEPRESSANTS, ANTIANXIETY AGENTS HOECHST MARION ROUSSEL, INC. (US) 1996-04-23 US disclosed
US-5292760-A 4-heteroaryl-1,3-benzodiazepines and 2-substituted-α-(heteroaryl)benzeneethanamines HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-03-08 US disclosed
EP-0322582-A2 4-Heteroaryl-1,3-Benzodiazepines and 2-substituted-alpha-(heteroaryl)benzeneethanamines, a process for their preparation and their use us medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-07-05 EP disclosed