SCHEMBL8945957

SCHEMBL8945957

CCCC1=Nc2ccccc2CC(c2sccc2C)N1C

nearest known ligand 0.31

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.31
PDE5A O76074 1/20 0.31
PDE6C P51160 1/20 0.31
PDE11A Q9HCR9 1/20 0.31
CTSD P07339 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8945738 0.98 HTT (0.30) HTTPDE5APDE6CPDE11A
SCHEMBL8946140 0.91 HTT (0.32) HTTPDE5APDE6CPDE11A
Hydrochloric Acid SCHEMBL8945828 0.89 HTT (0.31) HTTPDE5APDE6CPDE11A
SCHEMBL8945930 0.83 HTT (0.34) HTTPDE5ACTSD
SCHEMBL8945770 0.81 SLC6A2 (0.36) HTT
Hydrochloric Acid SCHEMBL8945896 0.81 HTT (0.33) HTTPDE5A
Hydrochloric Acid SCHEMBL8945853 0.81 SLC6A2 (0.36) HTT
SCHEMBL8945967 0.79 HRH4 (0.34) HTTPDE5A
SCHEMBL8945973 0.79 MEN1 (0.36) HTTPDE5A
SCHEMBL8946006 0.79 HTT (0.32) HTTPDE5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5510346-A ANTIDEPRESSANTS, ANTIANXIETY AGENTS HOECHST MARION ROUSSEL, INC. (US) 1996-04-23 US claimed
US-5510346-A ANTIDEPRESSANTS, ANTIANXIETY AGENTS HOECHST MARION ROUSSEL, INC. (US) 1996-04-23 US disclosed
US-5292760-A 4-heteroaryl-1,3-benzodiazepines and 2-substituted-α-(heteroaryl)benzeneethanamines HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-03-08 US disclosed