SCHEMBL8945973

SCHEMBL8945973

Cc1ccsc1C1Cc2ccccc2N=C(C2CC2)N1C

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
CYP2D6 P10635 1/20 0.36
RECQL P46063 1/20 0.36
BCHE P06276 2/20 0.33
ACHE P22303 1/20 0.33
HTT P42858 3/20 0.32
ALDH1A1 P00352 2/20 0.31
LMNA P02545 1/20 0.31
PDE5A O76074 2/20 0.31
KDM4E B2RXH2 2/20 0.31
HSD17B10 Q99714 1/20 0.31
GAA P10253 2/20 0.30
HPGD P15428 2/20 0.30
MAPT P10636 1/20 0.30
TDP1 Q9NUW8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8945930 0.85 HTT (0.34) MEN1KMT2ACYP2D6RECQLHTT
Hydrochloric Acid SCHEMBL8945896 0.83 HTT (0.33) MEN1KMT2ACYP2D6RECQLHTT
SCHEMBL8946140 0.81 HTT (0.32) MEN1KMT2AHTTALDH1A1PDE5A
SCHEMBL8945967 0.81 HRH4 (0.34) MEN1KMT2ABCHEHTTALDH1A1
SCHEMBL8946006 0.81 HTT (0.32) MEN1KMT2AHTTALDH1A1PDE5A
Hydrochloric Acid SCHEMBL8945964 0.80 HTT (0.32) HTTPDE5AKDM4EHSD17B10
Hydrochloric Acid SCHEMBL8945756 0.80 HRH4 (0.34) HTTPDE5AKDM4EHSD17B10
SCHEMBL8945957 0.79 HTT (0.31) HTTPDE5A
Hydrochloric Acid SCHEMBL8945828 0.79 HTT (0.31) HTTPDE5A
Hydrochloric Acid SCHEMBL8945738 0.77 HTT (0.30) HTTPDE5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5510346-A ANTIDEPRESSANTS, ANTIANXIETY AGENTS HOECHST MARION ROUSSEL, INC. (US) 1996-04-23 US disclosed
US-5292760-A 4-heteroaryl-1,3-benzodiazepines and 2-substituted-α-(heteroaryl)benzeneethanamines HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-03-08 US disclosed
EP-0322582-A2 4-Heteroaryl-1,3-Benzodiazepines and 2-substituted-alpha-(heteroaryl)benzeneethanamines, a process for their preparation and their use us medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-07-05 EP disclosed