SCHEMBL8946140

SCHEMBL8946140

CCC1=Nc2ccccc2CC(c2sccc2C)N1C

nearest known ligand 0.32

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.32
PDE5A O76074 3/20 0.32
PDE6C P51160 1/20 0.32
PDE11A Q9HCR9 1/20 0.32
KDM4E B2RXH2 2/20 0.31
HSD17B10 Q99714 1/20 0.31
GAA P10253 2/20 0.30
HPGD P15428 2/20 0.30
MEN1 O00255 1/20 0.30
ALDH1A1 P00352 1/20 0.30
MAPT P10636 1/20 0.30
KMT2A Q03164 1/20 0.30
TDP1 Q9NUW8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8945828 0.98 HTT (0.31) HTTPDE5APDE6CPDE11A
SCHEMBL8945957 0.91 HTT (0.31) HTTPDE5APDE6CPDE11A
Hydrochloric Acid SCHEMBL8945738 0.89 HTT (0.30) HTTPDE5APDE6CPDE11A
SCHEMBL8945910 0.86 ALDH1A1 (0.35) HTTKDM4EHSD17B10HPGDALDH1A1
SCHEMBL8945930 0.85 HTT (0.34) HTTPDE5AKDM4EHSD17B10GAA
SCHEMBL8946083 0.84 CRHR1 (0.33) HSD17B10MEN1KMT2A
SCHEMBL8945882 0.84
SCHEMBL8946007 0.84 ALDH1A1 (0.35) GAAALDH1A1
SCHEMBL8945811 0.84 ALDH1A1 (0.35) GAAALDH1A1
SCHEMBL8945744 0.83 KCNH2 (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5510346-A ANTIDEPRESSANTS, ANTIANXIETY AGENTS HOECHST MARION ROUSSEL, INC. (US) 1996-04-23 US claimed
EP-0322582-A2 4-Heteroaryl-1,3-Benzodiazepines and 2-substituted-alpha-(heteroaryl)benzeneethanamines, a process for their preparation and their use us medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-07-05 EP claimed
US-5510346-A ANTIDEPRESSANTS, ANTIANXIETY AGENTS HOECHST MARION ROUSSEL, INC. (US) 1996-04-23 US disclosed
US-5292760-A 4-heteroaryl-1,3-benzodiazepines and 2-substituted-α-(heteroaryl)benzeneethanamines HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-03-08 US disclosed
EP-0322582-A2 4-Heteroaryl-1,3-Benzodiazepines and 2-substituted-alpha-(heteroaryl)benzeneethanamines, a process for their preparation and their use us medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-07-05 EP disclosed