SCHEMBL8946003

SCHEMBL8946003

CCC1=Nc2ccccc2CC(c2ccc[nH]2)N1C

nearest known ligand 0.33

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.30
MEN1 O00255 1/20 0.30
RECQL P46063 1/20 0.30
KMT2A Q03164 1/20 0.30
MAOA P21397 1/20 0.30
MAOB P27338 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11270824 0.83 CHRNB2 (0.37) CYP2D6MEN1RECQLKMT2AMAOA
SCHEMBL8945976 0.81 ADRA1A (0.45) CYP2D6MEN1KMT2A
SCHEMBL8946144 0.80 CYP19A1 (0.34) CYP2D6RECQLKMT2AMAOAMAOB
SCHEMBL9583461 0.80 MAOA (0.40) MEN1KMT2AMAOAMAOB
SCHEMBL8945720 0.79
SCHEMBL9582044 0.79 NPY1R (0.36) MEN1RECQLKMT2A
SCHEMBL9582906 0.79 MAOB (0.41) MAOAMAOB
SCHEMBL9584219 0.79 MAOB (0.41) MEN1KMT2AMAOAMAOB
Water SCHEMBL8945782 0.79 CYP19A1 (0.33) CYP2D6KMT2AMAOAMAOB
Water SCHEMBL8945777 0.79 CYP19A1 (0.33) CYP2D6KMT2AMAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5510346-A ANTIDEPRESSANTS, ANTIANXIETY AGENTS HOECHST MARION ROUSSEL, INC. (US) 1996-04-23 US disclosed
US-5292760-A 4-heteroaryl-1,3-benzodiazepines and 2-substituted-α-(heteroaryl)benzeneethanamines HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-03-08 US disclosed
EP-0322582-A2 4-Heteroaryl-1,3-Benzodiazepines and 2-substituted-alpha-(heteroaryl)benzeneethanamines, a process for their preparation and their use us medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-07-05 EP disclosed