SCHEMBL8946004

SCHEMBL8946004

CNC(c1sccc1C)C(N)c1ccc(C(F)(F)F)cc1

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.31
KIF11 P52732 1/20 0.31
PDE2A O00408 1/20 0.31
GPR139 Q6DWJ6 1/20 0.30
MEN1 O00255 1/20 0.30
TP53 P04637 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2C9 P11712 1/20 0.30
TSHR P16473 1/20 0.30
CYP2C19 P33261 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9425307 0.85 PNMT (0.38) MEN1CYP1A2CYP3A4CYP2C9CYP2C19
Hydrochloric Acid SCHEMBL8946064 0.84 IDO1 (0.39)
SCHEMBL10588478 0.81 DPP4 (0.39) ALOX5
SCHEMBL9425406 0.72 ALOX5 (0.33) ALOX5CYP3A4
SCHEMBL13191168 0.70 CYP2C19 (0.52) KIF11PDE2AMEN1TP53CYP1A2
Hydrochloric Acid SCHEMBL8945996 0.69 DPP4 (0.34) ALOX5MEN1KMT2A
SCHEMBL15137434 0.68 KIF11 (0.46) KIF11PDE2ATSHR
SCHEMBL15670412 0.68 KIF11 (0.46) KIF11PDE2ATSHR
SCHEMBL10586629 0.67 CYP3A4 (0.37) ALOX5MEN1CYP3A4CYP2C9TSHR
SCHEMBL12569047 0.67 BCHE (0.42) KIF11PDE2ATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5292760-A 4-heteroaryl-1,3-benzodiazepines and 2-substituted-α-(heteroaryl)benzeneethanamines HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-03-08 US claimed
US-5510346-A ANTIDEPRESSANTS, ANTIANXIETY AGENTS HOECHST MARION ROUSSEL, INC. (US) 1996-04-23 US disclosed
US-5292760-A 4-heteroaryl-1,3-benzodiazepines and 2-substituted-α-(heteroaryl)benzeneethanamines HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-03-08 US disclosed
EP-0322582-A2 4-Heteroaryl-1,3-Benzodiazepines and 2-substituted-alpha-(heteroaryl)benzeneethanamines, a process for their preparation and their use us medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-07-05 EP disclosed