SCHEMBL9425307

SCHEMBL9425307

CNC(c1sccc1C)C(N)c1cccc(C(F)(F)F)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PNMT P11086 1/20 0.38
RAPGEF4 Q8WZA2 1/20 0.36
IDO1 P14902 1/20 0.36
TDO2 P48775 1/20 0.36
HTR2A P28223 1/20 0.36
HTR2C P28335 1/20 0.36
HTR2B P41595 1/20 0.36
KCNN4 O15554 1/20 0.36
DAO P14920 1/20 0.35
IDH2 P48735 1/20 0.34
AURKA O14965 1/20 0.34
OPRM1 P35372 2/20 0.33
OPRD1 P41143 2/20 0.33
OPRK1 P41145 2/20 0.33
OPRL1 P41146 2/20 0.33
CYP1A2 P05177 2/20 0.33
CYP3A4 P08684 2/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
CES2 O00748 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8946064 0.99 IDO1 (0.39) PNMTRAPGEF4IDO1TDO2HTR2A
SCHEMBL8946004 0.85 ALOX5 (0.31) CYP1A2CYP3A4CYP2C19MEN1CYP2C9
SCHEMBL9425406 0.81 ALOX5 (0.33) RAPGEF4IDO1TDO2CYP3A4SLC6A2
SCHEMBL10588478 0.80 DPP4 (0.39)
SCHEMBL30460663 0.77 PNMT (0.47) PNMTRAPGEF4IDO1TDO2KCNN4
SCHEMBL17465593 0.73 CES2 (0.50) PNMTIDO1TDO2HTR2AHTR2C
SCHEMBL29600944 0.73 CES2 (0.50) PNMTIDO1TDO2HTR2AHTR2C
SCHEMBL4524501 0.73 CES2 (0.50) PNMTIDO1TDO2HTR2AHTR2C
SCHEMBL2538654 0.73 CES2 (0.50) PNMTIDO1TDO2HTR2AHTR2C
SCHEMBL24017114 0.72 PNMT (0.59) PNMTIDO1TDO2HTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5292760-A 4-heteroaryl-1,3-benzodiazepines and 2-substituted-α-(heteroaryl)benzeneethanamines HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-03-08 US claimed