SCHEMBL8946008

SCHEMBL8946008

CC1=Nc2ccccc2CC(c2ccc(C)s2)N1C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 2/20 0.41
SLC6A2 P23975 1/20 0.41
SLC6A3 Q01959 1/20 0.41
DRD2 P14416 2/20 0.37
KMT2A Q03164 3/20 0.33
MEN1 O00255 2/20 0.33
CYP2D6 P10635 1/20 0.33
RECQL P46063 1/20 0.33
CTSD P07339 1/20 0.32
PDE5A O76074 1/20 0.31
PDE11A Q9HCR9 1/20 0.31
HRH4 Q9H3N8 1/20 0.31
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
HPGD P15428 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
HSD17B10 Q99714 1/20 0.31
HSD17B2 P37059 1/20 0.30
LMNA P02545 2/20 0.30
NPC1 O15118 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL10589042 0.99 SLC6A2 (0.40) SLC6A4SLC6A2SLC6A3DRD2KMT2A
SCHEMBL8945997 0.84 SLC6A2 (0.38) SLC6A4SLC6A2SLC6A3DRD2KMT2A
SCHEMBL8945774 0.82 SLC6A2 (0.40) SLC6A4SLC6A2SLC6A3KMT2AMEN1
Dazepinil SCHEMBL499286 0.80 CHRNB2 (0.40) KMT2AMEN1CYP2D6RECQLKDM4E
SCHEMBL8945994 0.78 HSD17B10 (0.34) KMT2AMEN1CYP2D6RECQLCTSD
SCHEMBL11266015 0.77 MAOA (0.43) KMT2AMEN1CYP2D6RECQLHPGD
SCHEMBL8945898 0.76 CYP19A1 (0.35) DRD2KMT2AMEN1CYP2D6RECQL
SCHEMBL8945930 0.76 HTT (0.34) DRD2KMT2AMEN1CYP2D6RECQL
SCHEMBL8945958 0.76 HRH4 (0.32) DRD2KMT2AMEN1CYP2D6RECQL
SCHEMBL11282542 0.75 MAOB (0.44) KMT2AMEN1KDM4EALDH1A1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5510346-A ANTIDEPRESSANTS, ANTIANXIETY AGENTS HOECHST MARION ROUSSEL, INC. (US) 1996-04-23 US claimed
US-5510346-A ANTIDEPRESSANTS, ANTIANXIETY AGENTS HOECHST MARION ROUSSEL, INC. (US) 1996-04-23 US disclosed
US-5292760-A 4-heteroaryl-1,3-benzodiazepines and 2-substituted-α-(heteroaryl)benzeneethanamines HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-03-08 US disclosed
EP-0322582-A2 4-Heteroaryl-1,3-Benzodiazepines and 2-substituted-alpha-(heteroaryl)benzeneethanamines, a process for their preparation and their use us medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-07-05 EP disclosed