SCHEMBL8945994

SCHEMBL8945994

CC1=Nc2ccccc2CC(c2ccsc2)N1C

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 2/20 0.34
TSHR P16473 1/20 0.34
ADORA2B P29275 3/20 0.34
NSD2 O96028 1/20 0.33
SMN1; SMN2 Q16637 3/20 0.32
LMNA P02545 1/20 0.32
MEN1 O00255 3/20 0.32
KMT2A Q03164 3/20 0.32
KDM4E B2RXH2 1/20 0.32
MAPT P10636 1/20 0.32
HRH4 Q9H3N8 1/20 0.32
HTT P42858 1/20 0.32
CYP2D6 P10635 1/20 0.31
RECQL P46063 1/20 0.31
CYP19A1 P11511 1/20 0.31
CTSD P07339 1/20 0.31
SIRT3 Q9NTG7 1/20 0.30
SIRT5 Q9NXA8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8945925 0.84 ADORA2B (0.32) ADORA2BHRH4
SCHEMBL8945923 0.84 HRH4 (0.35) HRH4
SCHEMBL8946148 0.84 ADORA2B (0.33) HSD17B10ADORA2BSMN1; SMN2LMNAMEN1
Dazepinil SCHEMBL499286 0.83 CHRNB2 (0.40) MEN1KMT2AKDM4ECYP2D6RECQL
Hydrochloric Acid SCHEMBL8945921 0.83 HRH4 (0.34) HRH4
Hydrochloric Acid SCHEMBL8945865 0.83 ADORA2B (0.32) ADORA2BSMN1; SMN2LMNAMEN1KMT2A
Hydrochloric Acid SCHEMBL8945951 0.82 ADORA2B (0.31) ADORA2B
SCHEMBL8945861 0.82 SMN1; SMN2 (0.32) ADORA2BSMN1; SMN2LMNAMEN1KMT2A
SCHEMBL8946123 0.81 OPRM1 (0.31) ADORA2BMEN1KMT2ACYP2D6RECQL
SCHEMBL11266015 0.81 MAOA (0.43) LMNAMEN1KMT2ACYP2D6RECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5510346-A ANTIDEPRESSANTS, ANTIANXIETY AGENTS HOECHST MARION ROUSSEL, INC. (US) 1996-04-23 US claimed
US-5510346-A ANTIDEPRESSANTS, ANTIANXIETY AGENTS HOECHST MARION ROUSSEL, INC. (US) 1996-04-23 US disclosed
US-5292760-A 4-heteroaryl-1,3-benzodiazepines and 2-substituted-α-(heteroaryl)benzeneethanamines HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-03-08 US disclosed
EP-0322582-A2 4-Heteroaryl-1,3-Benzodiazepines and 2-substituted-alpha-(heteroaryl)benzeneethanamines, a process for their preparation and their use us medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-07-05 EP disclosed