SCHEMBL8946028

SCHEMBL8946028

CC1=Nc2ccccc2CC(c2cn[nH]c2)N1C

nearest known ligand 0.33

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 3/20 0.33
CYP2D6 P10635 1/20 0.31
MEN1 O00255 1/20 0.31
RECQL P46063 1/20 0.31
KMT2A Q03164 1/20 0.31
ADORA2B P29275 1/20 0.30
ADORA1 P30542 1/20 0.30
ROCK2 O75116 1/20 0.30
CTSD P07339 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8946195 0.84 HSD11B1 (0.31) HSD11B1
Dazepinil SCHEMBL499286 0.82 CHRNB2 (0.40) CYP2D6MEN1RECQLKMT2A
SCHEMBL8946162 0.82 HSD11B1 (0.30) HSD11B1CTSD
SCHEMBL11266015 0.80 MAOA (0.43) CYP2D6MEN1RECQLKMT2A
SCHEMBL8945898 0.79 CYP19A1 (0.35) CYP2D6MEN1RECQLKMT2ACTSD
SCHEMBL8945889 0.78 CHRNB2 (0.48) MEN1KMT2A
SCHEMBL9582495 0.78 ALDH1A1 (0.41) MEN1RECQLKMT2A
SCHEMBL9583299 0.78 MAOB (0.42) KMT2A
SCHEMBL11282542 0.77 MAOB (0.44) MEN1KMT2A
SCHEMBL9583012 0.77 MEN1 (0.39) MEN1RECQLKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5510346-A ANTIDEPRESSANTS, ANTIANXIETY AGENTS HOECHST MARION ROUSSEL, INC. (US) 1996-04-23 US disclosed
US-5292760-A 4-heteroaryl-1,3-benzodiazepines and 2-substituted-α-(heteroaryl)benzeneethanamines HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-03-08 US disclosed
EP-0322582-A2 4-Heteroaryl-1,3-Benzodiazepines and 2-substituted-alpha-(heteroaryl)benzeneethanamines, a process for their preparation and their use us medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-07-05 EP disclosed