SCHEMBL8946053

SCHEMBL8946053

CNC(Cc1ccccc1OC)c1sccc1C

nearest known ligand 0.67

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.40
CYP2D6 P10635 3/20 0.40
CYP3A4 P08684 2/20 0.40
CYP2C19 P33261 2/20 0.40
CYP1A2 P05177 1/20 0.40
SLC6A2 P23975 1/20 0.39
SLC6A4 P31645 1/20 0.39
SLC6A3 Q01959 1/20 0.39
KCNH2 Q12809 1/20 0.39
ALDH1A1 P00352 1/20 0.38
GAA P10253 1/20 0.38
MAPT P10636 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8945983 0.99 CYP2D6 (0.42) HPGDCYP2D6CYP3A4CYP2C19CYP1A2
SCHEMBL9425146 0.82 CXCR1 (0.34) ALDH1A1MAPT
SCHEMBL8946017 0.81 ALOX5 (0.33) HPGDCYP3A4ALDH1A1
SCHEMBL8945768 0.81 HSPA5 (0.38) HPGDCYP2D6CYP3A4SLC6A2SLC6A4
Hydrochloric Acid SCHEMBL8946070 0.80 MAPT (0.39) HPGDCYP2D6CYP3A4SLC6A2SLC6A4
SCHEMBL8760252 0.77 TAAR1 (0.44) CYP2D6CYP2C19SLC6A2SLC6A4SLC6A3
Hydrochloric Acid SCHEMBL9482849 0.76 TAAR1 (0.43) CYP2D6CYP2C19
SCHEMBL8761001 0.75 MEN1 (0.41) HPGDALDH1A1MAPT
SCHEMBL8946175 0.74 MEN1 (0.34) CYP2D6ALDH1A1GAAMAPT
SCHEMBL8946095 0.74 ALDH1A1 (0.43) HPGDALDH1A1GAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5292760-A 4-heteroaryl-1,3-benzodiazepines and 2-substituted-α-(heteroaryl)benzeneethanamines HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-03-08 US claimed
US-5510346-A ANTIDEPRESSANTS, ANTIANXIETY AGENTS HOECHST MARION ROUSSEL, INC. (US) 1996-04-23 US disclosed
US-5292760-A 4-heteroaryl-1,3-benzodiazepines and 2-substituted-α-(heteroaryl)benzeneethanamines HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-03-08 US disclosed
EP-0322582-A2 4-Heteroaryl-1,3-Benzodiazepines and 2-substituted-alpha-(heteroaryl)benzeneethanamines, a process for their preparation and their use us medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-07-05 EP disclosed