SCHEMBL8946095

SCHEMBL8946095

CNC(Cc1ccccc1NC(C)=O)c1sccc1C

nearest known ligand 0.73

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.43
HPGD P15428 1/20 0.43
MAPT P10636 1/20 0.40
FEN1 P39748 1/20 0.39
TSHR P16473 1/20 0.38
MEN1 O00255 1/20 0.37
GAA P10253 1/20 0.37
KMT2A Q03164 1/20 0.37
CXCR1 P25024 1/20 0.37
CXCR2 P25025 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9425204 0.87 CETP (0.39) ALDH1A1MAPTMEN1GAAKMT2A
SCHEMBL9425146 0.86 CXCR1 (0.34) ALDH1A1MAPTKMT2ACXCR1CXCR2
SCHEMBL8945768 0.79 HSPA5 (0.38) ALDH1A1HPGDMAPTMEN1KMT2A
Hydrochloric Acid SCHEMBL8946070 0.78 MAPT (0.39) ALDH1A1HPGDMAPTMEN1KMT2A
SCHEMBL8946017 0.77 ALOX5 (0.33) ALDH1A1HPGDKMT2A
SCHEMBL9425074 0.76 MAPT (0.39) ALDH1A1MAPTMEN1GAAKMT2A
SCHEMBL9425072 0.76 CETP (0.38) ALDH1A1MAPTTSHRMEN1GAA
SCHEMBL8946053 0.74 HPGD (0.40) ALDH1A1HPGDMAPTGAA
SCHEMBL9425081 0.74 PGR (0.40) ALDH1A1HPGDMAPTMEN1GAA
SCHEMBL8761001 0.74 MEN1 (0.41) ALDH1A1HPGDMAPTTSHRMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5292760-A 4-heteroaryl-1,3-benzodiazepines and 2-substituted-α-(heteroaryl)benzeneethanamines HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-03-08 US claimed
US-5510346-A ANTIDEPRESSANTS, ANTIANXIETY AGENTS HOECHST MARION ROUSSEL, INC. (US) 1996-04-23 US disclosed
US-5292760-A 4-heteroaryl-1,3-benzodiazepines and 2-substituted-α-(heteroaryl)benzeneethanamines HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-03-08 US disclosed
EP-0322582-A2 4-Heteroaryl-1,3-Benzodiazepines and 2-substituted-alpha-(heteroaryl)benzeneethanamines, a process for their preparation and their use us medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-07-05 EP disclosed