SCHEMBL8946083

SCHEMBL8946083

CCC1=Nc2ccc(Br)cc2CC(c2sccc2C)N1C

nearest known ligand 0.33

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CRHR1 P34998 1/20 0.33
NPY1R P25929 1/20 0.32
MEN1 O00255 1/20 0.30
USP2 O75604 1/20 0.30
LMNA P02545 1/20 0.30
ALOX15 P16050 1/20 0.30
TSHR P16473 1/20 0.30
CASP1 P29466 1/20 0.30
CASP7 P55210 1/20 0.30
KMT2A Q03164 1/20 0.30
HSD17B10 Q99714 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8945910 0.89 ALDH1A1 (0.35) CRHR1LMNAALOX15TSHRHSD17B10
SCHEMBL8945882 0.87
SCHEMBL8946007 0.87 ALDH1A1 (0.35) CRHR1TSHR
SCHEMBL8946140 0.84 HTT (0.32) MEN1KMT2AHSD17B10
Hydrochloric Acid SCHEMBL8945828 0.82 HTT (0.31)
SCHEMBL8945811 0.80 ALDH1A1 (0.35) CRHR1LMNATSHR
SCHEMBL8945957 0.76 HTT (0.31)
Hydrochloric Acid SCHEMBL8945738 0.74 HTT (0.30)
SCHEMBL9582044 0.69 NPY1R (0.36) NPY1RMEN1LMNAKMT2A
SCHEMBL8945744 0.68 KCNH2 (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5510346-A ANTIDEPRESSANTS, ANTIANXIETY AGENTS HOECHST MARION ROUSSEL, INC. (US) 1996-04-23 US disclosed
US-5292760-A 4-heteroaryl-1,3-benzodiazepines and 2-substituted-α-(heteroaryl)benzeneethanamines HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-03-08 US disclosed
EP-0322582-A2 4-Heteroaryl-1,3-Benzodiazepines and 2-substituted-alpha-(heteroaryl)benzeneethanamines, a process for their preparation and their use us medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-07-05 EP disclosed