SCHEMBL8945910

SCHEMBL8945910

CCC1=Nc2ccc(C)cc2CC(c2sccc2C)N1C

nearest known ligand 0.35

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.35
LMNA P02545 2/20 0.35
KDM4E B2RXH2 1/20 0.35
TP53 P04637 1/20 0.35
MAPT P10636 1/20 0.35
HPGD P15428 1/20 0.35
ALOX15 P16050 1/20 0.35
TSHR P16473 1/20 0.35
HSD17B10 Q99714 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
PDE3B Q13370 1/20 0.34
PDE3A Q14432 1/20 0.34
CRHR1 P34998 1/20 0.31
HTT P42858 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8946083 0.89 CRHR1 (0.33) LMNAALOX15TSHRHSD17B10CRHR1
SCHEMBL8946140 0.86 HTT (0.32) ALDH1A1KDM4EMAPTHPGDHSD17B10
Hydrochloric Acid SCHEMBL8945828 0.84 HTT (0.31) HTT
SCHEMBL8945811 0.82 ALDH1A1 (0.35) ALDH1A1LMNATP53TSHRCRHR1
SCHEMBL8945957 0.77 HTT (0.31) HTT
Hydrochloric Acid SCHEMBL8945738 0.76 HTT (0.30) HTT
SCHEMBL8945930 0.71 HTT (0.34) ALDH1A1LMNAKDM4ETP53MAPT
SCHEMBL8945744 0.70 KCNH2 (0.31)
Hydrochloric Acid SCHEMBL8945896 0.69 HTT (0.33) ALDH1A1KDM4EMAPTHPGDHSD17B10
SCHEMBL9582776 0.69 DRD2 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5510346-A ANTIDEPRESSANTS, ANTIANXIETY AGENTS HOECHST MARION ROUSSEL, INC. (US) 1996-04-23 US disclosed
US-5292760-A 4-heteroaryl-1,3-benzodiazepines and 2-substituted-α-(heteroaryl)benzeneethanamines HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-03-08 US disclosed
EP-0322582-A2 4-Heteroaryl-1,3-Benzodiazepines and 2-substituted-alpha-(heteroaryl)benzeneethanamines, a process for their preparation and their use us medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-07-05 EP disclosed