SCHEMBL8946086

SCHEMBL8946086

CNC(Cc1ccc(N)cc1)c1csc(Cl)n1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
RAD52 P43351 2/20 0.41
SOAT1 P35610 1/20 0.32
PTPRB P23467 2/20 0.32
ALDH1A1 P00352 1/20 0.32
CYP3A4 P08684 1/20 0.32
TSHR P16473 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
BACE1 P56817 1/20 0.32
ESR1 P03372 1/20 0.31
CYP19A1 P11511 1/20 0.30
NPC1 O15118 1/20 0.30
RAB9A P51151 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24534131 0.82 PTPRB (0.41) RAD52SOAT1PTPRBALDH1A1CYP3A4
SCHEMBL24534166 0.77 PTPRB (0.47) RAD52PTPRBTDP1NPC1RAB9A
SCHEMBL24534181 0.73 PTPRB (0.41) PTPRBALDH1A1NPC1RAB9A
SCHEMBL21914932 0.70 PTPRB (0.47) PTPRBBACE1NPC1RAB9A
SCHEMBL22267911 0.69 CCR3 (0.39) RAD52SOAT1PTPRBALDH1A1CYP3A4
SCHEMBL19257745 0.69 CCR3 (0.39) RAD52SOAT1PTPRBALDH1A1CYP3A4
SCHEMBL7182179 0.68 ALDH1A1 (0.50) ALDH1A1CYP3A4TSHRTDP1
SCHEMBL24534174 0.67 MEN1 (0.49) PTPRBALDH1A1CYP3A4TDP1CYP19A1
SCHEMBL21914203 0.67 PTPRB (0.48) RAD52SOAT1PTPRBBACE1
SCHEMBL24534145 0.64 RAB9A (0.41) PTPRBALDH1A1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5510346-A ANTIDEPRESSANTS, ANTIANXIETY AGENTS HOECHST MARION ROUSSEL, INC. (US) 1996-04-23 US disclosed
US-5292760-A 4-heteroaryl-1,3-benzodiazepines and 2-substituted-α-(heteroaryl)benzeneethanamines HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-03-08 US disclosed
EP-0322582-A2 4-Heteroaryl-1,3-Benzodiazepines and 2-substituted-alpha-(heteroaryl)benzeneethanamines, a process for their preparation and their use us medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-07-05 EP disclosed