SCHEMBL8946094

SCHEMBL8946094

CNC(Cc1ccccc1N)c1ccn(C)c1

nearest known ligand 0.50

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.30
OPRK1 P41145 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9001661 0.80 ALDH1A1 (0.42) SIGMAR1
Hydrochloric Acid SCHEMBL9582763 0.79 ALDH1A1 (0.41) SIGMAR1
Hydrochloric Acid SCHEMBL9001659 0.79 ALDH1A1 (0.41) SIGMAR1
SCHEMBL10565227 0.76 GAA (0.38)
SCHEMBL8946113 0.75 MEN1 (0.33) SIGMAR1
SCHEMBL8945887 0.75 IDO1 (0.36)
SCHEMBL9583350 0.75 ALDH1A1 (0.37)
Hydrochloric Acid SCHEMBL9582349 0.75 TDP1 (0.37)
SCHEMBL8945848 0.75 CYP3A4 (0.42)
SCHEMBL9583244 0.72 ALDH1A1 (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5510346-A ANTIDEPRESSANTS, ANTIANXIETY AGENTS HOECHST MARION ROUSSEL, INC. (US) 1996-04-23 US disclosed
US-5292760-A 4-heteroaryl-1,3-benzodiazepines and 2-substituted-α-(heteroaryl)benzeneethanamines HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-03-08 US disclosed
EP-0322582-A2 4-Heteroaryl-1,3-Benzodiazepines and 2-substituted-alpha-(heteroaryl)benzeneethanamines, a process for their preparation and their use us medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-07-05 EP disclosed