SCHEMBL8945887

SCHEMBL8945887

CNC(Cc1ccccc1N)c1ccsc1

nearest known ligand 0.58

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.36
TDO2 P48775 1/20 0.36
SLC6A2 P23975 2/20 0.34
SLC6A4 P31645 2/20 0.34
ADRB3 P13945 1/20 0.32
ALOX5 P09917 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
SLC6A3 Q01959 1/20 0.31
KCNH2 Q12809 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9001661 0.81 ALDH1A1 (0.42)
Hydrochloric Acid SCHEMBL9001659 0.80 ALDH1A1 (0.41)
Hydrochloric Acid SCHEMBL9582763 0.80 ALDH1A1 (0.41)
SCHEMBL10565227 0.77 GAA (0.38) SLC6A4
SCHEMBL9583350 0.76 ALDH1A1 (0.37) SLC6A2SLC6A4CYP3A4CYP2D6SLC6A3
Hydrochloric Acid SCHEMBL9582349 0.76 TDP1 (0.37) CYP3A4
SCHEMBL8945848 0.76 CYP3A4 (0.42) SLC6A2SLC6A4CYP3A4SLC6A3
SCHEMBL8945940 0.75 KDM4E (0.31) CYP3A4
SCHEMBL8946094 0.75 SIGMAR1 (0.30)
SCHEMBL8945903 0.75 LTA4H (0.36) SLC6A2SLC6A4CYP3A4CYP2D6SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5292760-A 4-heteroaryl-1,3-benzodiazepines and 2-substituted-α-(heteroaryl)benzeneethanamines HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-03-08 US claimed
US-5510346-A ANTIDEPRESSANTS, ANTIANXIETY AGENTS HOECHST MARION ROUSSEL, INC. (US) 1996-04-23 US disclosed
US-5292760-A 4-heteroaryl-1,3-benzodiazepines and 2-substituted-α-(heteroaryl)benzeneethanamines HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-03-08 US disclosed
EP-0322582-A2 4-Heteroaryl-1,3-Benzodiazepines and 2-substituted-alpha-(heteroaryl)benzeneethanamines, a process for their preparation and their use us medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-07-05 EP disclosed