SCHEMBL8946181

SCHEMBL8946181

CS(=O)(=O)N1CC(=O)Sc2ccccc2C1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 1/20 0.40
RYR2 Q92736 1/20 0.37
ALDH1A1 P00352 5/20 0.37
KDM4E B2RXH2 2/20 0.37
HPGD P15428 2/20 0.37
ESR1 P03372 1/20 0.35
ESR2 Q92731 1/20 0.35
TSHR P16473 3/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
KMT2A Q03164 4/20 0.34
MEN1 O00255 3/20 0.34
HTT P42858 1/20 0.34
ATM Q13315 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
PRMT5 O14744 1/20 0.33
WDR77 Q9BQA1 1/20 0.33
MAPK1 P28482 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1266336 0.78 ESR1 (0.49) ALDH1A1ESR1ESR2TSHRKMT2A
SCHEMBL7559963 0.74 RYR2 (0.63) KDM1ARYR2ALDH1A1ESR1ESR2
SCHEMBL16503316 0.71 KMT2A (0.44) ALDH1A1KDM4EESR1ESR2TSHR
SCHEMBL6677893 0.67 BRD4 (0.46) RYR2ALDH1A1KDM4EHPGDKMT2A
SCHEMBL2103706 0.67 KMT2A (0.64) ESR1ESR2TSHRNPSR1KMT2A
SCHEMBL1498003 0.67 ALDH1A1 (0.59) RYR2ALDH1A1KDM4EHPGDKMT2A
Sulfuric Acid SCHEMBL30114767 0.66 CES1 (0.41) ALDH1A1KDM4EHPGDTSHRNPC1
SCHEMBL6238887 0.65 ALDH1A1 (0.47) ALDH1A1KDM4EHPGDTSHRNPC1
SCHEMBL29836089 0.65 ALDH1A1 (0.47) ALDH1A1KDM4EHPGDTSHRNPC1
SCHEMBL11633335 0.65 MAOA (0.50) KDM1AALDH1A1KDM4EHPGDTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5580866-A Therapeutic 1,4-thiazepines THE BOOTS COMPANY PLC (GB) 1996-12-03 US claimed