SCHEMBL8946329

SCHEMBL8946329

COc1cc(C(C)C)c2c(c1)[C@H]1Cc3ccccc3[C@@]1(C)N2

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 5/20 0.35
LPAR1 Q92633 5/20 0.35
HTR2A P28223 1/20 0.34
HTR2C P28335 1/20 0.34
HTR2B P41595 1/20 0.34
ALDH1A1 P00352 1/20 0.33
MEN1 O00255 1/20 0.33
CYP2D6 P10635 1/20 0.33
ALOX15 P16050 1/20 0.33
CYP2C19 P33261 1/20 0.33
KMT2A Q03164 1/20 0.33
GRIN2D O15399 1/20 0.33
GRIN3B O60391 1/20 0.33
BCHE P06276 1/20 0.33
CHRM5 P08912 1/20 0.33
TSHR P16473 1/20 0.33
ALOX12 P18054 1/20 0.33
NFKB1 P19838 1/20 0.33
MAPK1 P28482 1/20 0.33
PRCP P42785 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8946333 1.00 CYP3A4 (0.35) CYP3A4LPAR1HTR2AHTR2CHTR2B
SCHEMBL8946323 1.00 CYP3A4 (0.35) CYP3A4LPAR1HTR2AHTR2CHTR2B
SCHEMBL8946537 0.85 HTR2A (0.36) CYP3A4HTR2AHTR2CHTR2BALDH1A1
SCHEMBL8946545 0.85 HTR2A (0.36) CYP3A4HTR2AHTR2CHTR2BALDH1A1
SCHEMBL8946539 0.85 HTR2A (0.36) CYP3A4HTR2AHTR2CHTR2BALDH1A1
SCHEMBL9844749 0.73 HTR2A (0.34) HTR2AHTR2CHTR2BALDH1A1
SCHEMBL9844752 0.73 HTR2A (0.34) HTR2AHTR2CHTR2BALDH1A1
SCHEMBL9844750 0.73 HTR2A (0.34) HTR2AHTR2CHTR2BALDH1A1
SCHEMBL8946653 0.71 MAOA (0.32) HTR2AHTR2CHTR2BALDH1A1MEN1
SCHEMBL8946661 0.71 MAOA (0.32) HTR2AHTR2CHTR2BALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5516788-A TREATMENT OF ATHEROSCLEROSIS; ANTIISCHEMIC, ANTICARCINOGENIC AGENTS; ANTICOAGULANTS UNIVERSITY OF BATH (GB) 1996-05-14 US disclosed
EP-0409410-B1 Indenoindole compounds UNIV BATH (GB) 1996-03-20 EP disclosed
EP-0409410-A1 Indenoindole compounds UNIVERSITY OF BATH (GB) 1991-01-23 EP disclosed