SCHEMBL8946500

SCHEMBL8946500

CC(C)c1ccc2c(c1)C1Cc3ccccc3C1N2C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
LMNA P02545 1/20 0.43
MAPT P10636 1/20 0.43
HPGD P15428 1/20 0.43
MAPK1 P28482 1/20 0.43
HTT P42858 1/20 0.43
OPRM1 P35372 4/20 0.36
OPRK1 P41145 2/20 0.36
HSP90AA1 P07900 1/20 0.33
HSP90AB1 P08238 1/20 0.33
NR1H3 Q13133 1/20 0.33
CHRNB2 P17787 2/20 0.33
CHRNA4 P43681 2/20 0.33
HTR2A P28223 2/20 0.33
KCNH2 Q12809 2/20 0.31
ADRA2A P08913 1/20 0.31
ADRA2B P18089 1/20 0.31
ADRA2C P18825 1/20 0.31
SLC6A2 P23975 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8946497 1.00 KDM4E (0.43) KDM4EALDH1A1LMNAMAPTHPGD
SCHEMBL8946506 1.00 KDM4E (0.43) KDM4EALDH1A1LMNAMAPTHPGD
SCHEMBL8946433 0.82 SLC6A2 (0.40) KDM4EALDH1A1MAPTOPRM1CHRNB2
SCHEMBL8946437 0.82 SLC6A2 (0.40) KDM4EALDH1A1MAPTOPRM1CHRNB2
SCHEMBL8946442 0.82 SLC6A2 (0.40) KDM4EALDH1A1MAPTOPRM1CHRNB2
SCHEMBL10380873 0.81 HPGD (0.55) KDM4EALDH1A1LMNAMAPTHPGD
SCHEMBL8946743 0.81 ADRA2A (0.41) OPRM1OPRK1CHRNB2CHRNA4HTR2A
SCHEMBL8946720 0.81 ADRA2A (0.41) OPRM1OPRK1CHRNB2CHRNA4HTR2A
SCHEMBL8946747 0.81 ADRA2A (0.41) OPRM1OPRK1CHRNB2CHRNA4HTR2A
SCHEMBL24300090 0.81 OPRM1 (0.41) OPRM1OPRK1HTR2ASLC6A2HTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5516788-A TREATMENT OF ATHEROSCLEROSIS; ANTIISCHEMIC, ANTICARCINOGENIC AGENTS; ANTICOAGULANTS UNIVERSITY OF BATH (GB) 1996-05-14 US disclosed
EP-0409410-B1 Indenoindole compounds UNIV BATH (GB) 1996-03-20 EP disclosed
WO-1990015799-A1 INDENOINDOLE COMPOUNDS II UNIVERSITY OF BATH (GB) 1990-12-27 WO disclosed